Target Details
| UniProt AC | O76083 |
|---|---|
| Gene Symbol | PDE9A |
| Protein Name | High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) |
Summary
- Multi-target molecules 62
- Clinical molecules 0
- Avg pChEMBL 7.95
KEGG Pathways (2)
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJLHNYPXKZJKLV
|
10.0 | IC50 | 24 | — | |
KXCOKRBRUWINCT
|
9.9 | IC50 | 24 | — | |
KPFFPWNKWSYQFT
|
9.8 | IC50 | 24 | — | |
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
UBBCZBKJYNXHGT
|
9.2 | IC50 | 3 | — | |
GGDJPBJMQBKBTC
|
9.1 | IC50 | 2 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
HACIQJUXQZLQEN
|
9.0 | IC50 | 2 | — | |
JPRBQBBNWFDFSU
|
8.9 | IC50 | 2 | — | |
BRMLQSDHYPTXMV
|
8.8 | IC50 | 2 | — | |
SNCRCEGCQVMUBS
|
8.7 | IC50 | 3 | — | |
SNCRCEGCQVMUBS
|
8.7 | IC50 | 2 | — | |
FVOYQCUKGQGDKH
|
8.7 | IC50 | 2 | — | |
UBBCZBKJYNXHGT
|
8.5 | IC50 | 2 | — | |
RHYNVXDLIQWYAD
|
8.5 | IC50 | 2 | — | |
YZDGDEYKWUSLMC
|
8.4 | IC50 | 2 | — | |
FVSFTKVUXVUPHI
|
8.3 | IC50 | 2 | — | |
VGTCMYGKGIMPKU
|
8.3 | IC50 | 2 | — | |
NGJKWXIPEUHCJA
|
8.2 | IC50 | 2 | — | |
IJNPZLODDCNVFR
|
8.2 | IC50 | 2 | — | |
UJQKNBFBUSXTSO
|
8.2 | IC50 | 2 | — | |
GJXGHHNPNGRGBH
|
8.1 | IC50 | 2 | — | |
UORHIBXCPUHXFY
|
8.1 | IC50 | 4 | — | |
ZRIDRENRJOMKEQ
|
8.1 | IC50 | 3 | — | |
GNDFTZVYDQRFCD
|
8.1 | Ki | 2 | — | |
QEJJXMNBAFWGJK
|
8.0 | IC50 | 3 | — | |
FBJORBQVOXYGJP
|
8.0 | IC50 | 2 | — | |
FIUCLBJMUGCQTF
|
8.0 | IC50 | 8 | — | |
LLIYAZFYRUESNK
|
8.0 | IC50 | 2 | — | |
LRZBUWUBWWKUDL
|
8.0 | IC50 | 2 | — | |
JSAHYUSOARFYAP
|
7.9 | IC50 | 2 | — | |
GXVMSDLIIROULV
|
7.8 | IC50 | 2 | — | |
FIUCLBJMUGCQTF
|
7.8 | IC50 | 2 | — | |
VBTOPTREEDAWSQ
|
7.8 | IC50 | 2 | — | |
YFLRWBCQIACXIL
|
7.8 | IC50 | 2 | — | |
KKFKLLKJGDFZBA
|
7.7 | IC50 | 2 | — | |
FHBANDDJQJAZOQ
|
7.7 | IC50 | 2 | — | |
XFWJNKPDHNMLIO
|
7.5 | IC50 | 2 | — | |
HJXAXXUTIBEZHT
|
7.5 | IC50 | 2 | — | |
GYKSGQMBFSLYGY
|
7.4 | IC50 | 2 | — | |
KKFKLLKJGDFZBA
|
7.3 | IC50 | 2 | — | |
FFPXPXOAFQCNBS
|
7.3 | IC50 | 2 | — | |
RCKCFOKBILAFJF
|
7.2 | IC50 | 2 | — | |
FIUCLBJMUGCQTF
|
7.2 | IC50 | 3 | — | |
INDDKWKJTWMRQK
|
7.2 | IC50 | 3 | — | |
STXRQVNFUFZKSJ
|
7.2 | IC50 | 2 | — | |
UWLURVWZRQXQEM
|
7.2 | IC50 | 3 | — |