Target Details
| UniProt AC | O75914 |
|---|---|
| Gene Symbol | PAK3 |
| Protein Name | Serine/threonine-protein kinase PAK 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00786 (PBD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 35
- Clinical molecules 8
- Avg pChEMBL 6.92
KEGG Pathways (11)
Associated Diseases (1)
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.3 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
8.2 | Kd | 213 | — | |
WINHZLLDWRZWRT
|
7.8 | Kd | 201 | Yes | |
QQWUGDVOUVUTOY
|
7.5 | Kd | 231 | Yes | |
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
GUERACYCGKAFOU
|
7.3 | IC50 | 3 | — | |
HISDSBBMGJUNCI
|
7.2 | IC50 | 3 | — | |
FTGUWURNNBVUBC
|
7.2 | IC50 | 3 | — | |
AKBMXDMYBOYBBK
|
7.2 | IC50 | 3 | — | |
GHYZGSZITPRQRZ
|
7.2 | IC50 | 3 | — | |
WFVHHGNMKJUPFM
|
7.1 | IC50 | 3 | — | |
WFVHHGNMKJUPFM
|
7.0 | IC50 | 3 | — | |
AYCPARAPKDAOEN
|
7.0 | IC50 | 73 | — | |
MOSKATHMXWSZTQ
|
7.0 | IC50 | 16 | Yes | |
SGUZXWKWTMWMCR
|
6.9 | IC50 | 4 | — | |
PVZRBQHDDWNKDW
|
6.9 | IC50 | 3 | — | |
QKNBRNSGPNCARD
|
6.8 | IC50 | 9 | — | |
AAMUKYFUFDUBDC
|
6.8 | IC50 | 3 | — | |
QWFHISYETQDHDU
|
6.8 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 91 | Yes | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — | |
UEKXGVNKFSFQPH
|
6.7 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
6.7 | Kd | 165 | Yes | |
GTAKUJFUJVMIPM
|
6.6 | IC50 | 3 | — | |
WTEGSNARHOVIJM
|
6.6 | IC50 | 3 | — | |
DTIPYTJPPYYCBX
|
6.6 | IC50 | 3 | — | |
WFVHHGNMKJUPFM
|
6.6 | IC50 | 3 | — | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
HKJCMFRABFUAJX
|
6.4 | IC50 | 9 | — | |
YYLKKYCXAOBSRM
|
6.3 | Kd | 191 | — | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
PIQCTGMSNWUMAF
|
6.1 | Kd | 137 | Yes | |
YABJJWZLRMPFSI
|
6.1 | Kd | 34 | — | |
WFVHHGNMKJUPFM
|
6.1 | IC50 | 3 | — |