Target Details
| UniProt AC | O75716 |
|---|---|
| Gene Symbol | STK16 |
| Protein Name | Serine/threonine-protein kinase 16 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 456
- Clinical molecules 402
- Avg pChEMBL 7.28
Active Molecules (456)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJIAQDJKSXQLIT
|
6.3 | Kd | 38 | — | |
DORZPJWJOBMQKC
|
6.2 | IC50 | 9 | — | |
HMUZWZQGRIJSCT
|
6.2 | pIC50 | 2 | Yes | |
DVKYBHNNFVMHIN
|
6.2 | pIC50 | 3 | Yes | |
KEZAFIAURWAGLZ
|
6.2 | pIC50 | 3 | Yes | |
NFCAJLCVTMPSFF
|
6.2 | pIC50 | 2 | Yes | |
QVWIVWPIJUYRRF
|
6.2 | pIC50 | 8 | Yes | |
FATFDRYYCYZBQB
|
6.2 | pIC50 | 5 | Yes | |
ZGTHJDQZGGIPLL
|
6.2 | pIC50 | 5 | Yes | |
AIQJXTOEZSDXHV
|
6.2 | pIC50 | 3 | Yes | |
HZGUNBBYCUIOFD
|
6.2 | pIC50 | 2 | Yes | |
CIWJUMXZAYFUEI
|
6.2 | pIC50 | 2 | Yes | |
DCBGVRDAEOIKPQ
|
6.2 | pIC50 | 5 | Yes | |
WKBCIZTZDKGBEO
|
6.2 | pIC50 | 3 | Yes | |
ZYYNXHSAMWEIKK
|
6.2 | pIC50 | 4 | Yes | |
KSAUSYLGKMZHPT
|
6.2 | pIC50 | 3 | Yes | |
CTNPALGJUAXMMC
|
6.1 | Kd | 151 | — | |
ZCGDFAQAYLXLJV
|
6.1 | pIC50 | 2 | Yes | |
IFTCXKUSJMWVRD
|
6.1 | pIC50 | 7 | Yes | |
NMULSNNATHYGPZ
|
6.1 | pIC50 | 3 | Yes | |
DPYASQWYHILTBI
|
6.1 | pIC50 | 6 | Yes | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
SJHYJOUKZAHFOM
|
6.1 | pIC50 | 3 | Yes | |
ILOAUSWXRCKWFH
|
6.1 | pIC50 | 3 | Yes | |
WKDACQVEJIVHMZ
|
6.1 | Kd | 46 | — | |
FWLMVFUGMHIOAA
|
6.0 | Kd | 26 | — | |
IGRYEDIMNMEBBU
|
6.0 | IC50 | 9 | — | |
VFGWASLDLFTQPZ
|
6.0 | pIC50 | 6 | Yes | |
IYTGPPNUOLLGBE
|
6.0 | pIC50 | 2 | Yes | |
GASPHORHXIOCBB
|
6.0 | pIC50 | 4 | Yes | |
ZNGNLXZBVWXEKM
|
6.0 | pIC50 | 2 | Yes | |
GEUNWTZTVWNSTN
|
6.0 | pIC50 | 3 | Yes | |
IMQVBCRZLIQNPG
|
6.0 | pIC50 | 5 | Yes | |
XQWUFPUUHVVAIM
|
6.0 | pIC50 | 2 | Yes | |
CVFYLUGNOLKEFO
|
6.0 | IC50 | 7 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JOAWBRMGMMCJGS
|
6.0 | pIC50 | 4 | Yes | |
TXXYVBLFLGPQOR
|
6.0 | pIC50 | 5 | Yes | |
BMGGDZTXJBWQCN
|
Clinical | TTD_MultiTarget | 2 | Yes | |
CQRFXINTEFATOH
|
Clinical | TTD_MultiTarget | 2 | Yes | |
CQRFXINTEFATOH
|
Clinical | TTD_MultiTarget | 2 | Yes | |
DUPIINAVKMGMHG
|
Clinical | TTD_MultiTarget | 2 | Yes | |
FLGQTDLHJSQLIG
|
Clinical | TTD_MultiTarget | 2 | Yes | |
FQCMIMYFHWLFTJ
|
Clinical | TTD_MultiTarget | 2 | Yes | |
HLILQABBLFGERM
|
Clinical | TTD_MultiTarget | 6 | Yes | |
HVNQYDHDQBJAAH
|
Clinical | TTD_MultiTarget | 2 | Yes | |
JPOSFPUHBHRUAX
|
Clinical | TTD_MultiTarget | 40 | Yes | |
LDKHTALMQVJDPD
|
Clinical | TTD_MultiTarget | 4 | Yes | |
NCSQDKMOKNQGSG
|
Clinical | TTD_MultiTarget | 3 | Yes | |
NQVSRBQAHLEDFP
|
Clinical | TTD_MultiTarget | 3 | Yes |