Target Details
| UniProt AC | O75716 |
|---|---|
| Gene Symbol | STK16 |
| Protein Name | Serine/threonine-protein kinase 16 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 456
- Clinical molecules 402
- Avg pChEMBL 7.28
Active Molecules (456)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JTGMDPHLGBACAV
|
6.7 | pIC50 | 5 | Yes | |
LCNZVWVKIFPDPM
|
6.7 | pIC50 | 3 | Yes | |
XLJHIFICPVNHJG
|
6.7 | pIC50 | 2 | Yes | |
PCWVNRZWJPOOHP
|
6.7 | pIC50 | 3 | Yes | |
CCIYHYFLYIQCJR
|
6.7 | pIC50 | 3 | Yes | |
HCTOHQBQSMBFHY
|
6.7 | pIC50 | 2 | Yes | |
INTMVZKGQXMUML
|
6.7 | Ki | 3 | — | |
JCXULQAGBNATOH
|
6.7 | pIC50 | 3 | Yes | |
JVXJMEFHHQBIIG
|
6.7 | pIC50 | 3 | Yes | |
RGGYJEYZTPRESN
|
6.7 | pIC50 | 6 | Yes | |
OPSVHJZYWJYWSU
|
6.6 | pIC50 | 3 | Yes | |
RPGZQOOZHIEPJW
|
6.6 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
6.6 | Kd | 18 | — | |
XZDKAVSSXNBWNJ
|
6.6 | pIC50 | 5 | Yes | |
DWCZEZXJZXJTHE
|
6.6 | pIC50 | 6 | Yes | |
HBGNZQRVHBIHPS
|
6.6 | pIC50 | 6 | Yes | |
HFTUUUTZQAVFBK
|
6.6 | pIC50 | 3 | Yes | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 408 | — | |
YLVDJOXELSCRPM
|
6.6 | Ki | 3 | — | |
FKLCPPPITVKULK
|
6.6 | pIC50 | 3 | Yes | |
WINHZLLDWRZWRT
|
6.6 | Kd | 201 | Yes | |
MZWALFBOTNMRTP
|
6.6 | pIC50 | 7 | Yes | |
DIGPGAQNZZWPSG
|
6.6 | pIC50 | 3 | Yes | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 213 | — | |
PRASIGARSOSUQT
|
6.6 | pIC50 | 11 | Yes | |
UCBIQZUJJSVQHL
|
6.6 | Ki | 8 | — | |
XXSQNJQHHHVCBG
|
6.6 | pIC50 | 7 | Yes | |
DQJRSRINKOLTGU
|
6.6 | pIC50 | 2 | Yes | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 91 | Yes | |
GVMDVMPNOAVKJR
|
6.5 | pIC50 | 26 | Yes | |
HMCLAGIMLMMAEF
|
6.5 | pIC50 | 3 | Yes | |
KGXUJVJQAAUOTC
|
6.5 | pIC50 | 2 | Yes | |
XTWXMJDVQOEURD
|
6.5 | pIC50 | 3 | Yes | |
MCYCSSJHDPRHBZ
|
6.5 | Ki | 4 | — | |
RSIMWZIJZCXPJV
|
6.5 | pIC50 | 3 | Yes | |
XOUJEIXPUNKLEG
|
6.5 | IC50 | 3 | — | |
UJBJAMOSBBJZBK
|
6.5 | pIC50 | 6 | Yes | |
GFDMYTNCMHUIAT
|
6.5 | pIC50 | 2 | Yes | |
IMYVCWQAHSYYOO
|
6.5 | pIC50 | 2 | Yes | |
NKCMEGZSWOVKIL
|
6.5 | Ki | 3 | — | |
WHFRCTYFOGGZAU
|
6.5 | pIC50 | 2 | Yes | |
CZVVMRNEBRFYTL
|
6.5 | pIC50 | 9 | Yes | |
HVNQYDHDQBJAAH
|
6.5 | pIC50 | 3 | Yes | |
HSMLVQPVLGLUCI
|
6.5 | pIC50 | 2 | Yes | |
HJDMEPOCEJXNJU
|
6.5 | Ki | 3 | — | |
CULXCGPBYYEBGM
|
6.5 | pIC50 | 2 | Yes | |
SSHDKAJDJAVHAF
|
6.5 | pIC50 | 8 | Yes | |
FMMQGWSMYANLDD
|
6.5 | pIC50 | 3 | Yes | |
GXQWWDBZTZLIAJ
|
6.5 | Ki | 3 | — |