Target Details
| UniProt AC | O75716 |
|---|---|
| Gene Symbol | STK16 |
| Protein Name | Serine/threonine-protein kinase 16 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 456
- Clinical molecules 402
- Avg pChEMBL 7.28
Active Molecules (456)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OGNYUTNQZVRGMN
|
7.0 | pIC50 | 16 | Yes | |
QSIAXFKUFXOHHK
|
7.0 | pIC50 | 5 | Yes | |
SCANZEHBHPIJEQ
|
7.0 | pIC50 | 2 | Yes | |
YUPOZANDWNEEJQ
|
7.0 | pIC50 | 3 | Yes | |
DYTKVFHLKPDNRW
|
7.0 | pIC50 | 23 | Yes | |
YIQYJKSVIIKEJE
|
7.0 | pIC50 | 2 | Yes | |
YLJSAFSDGFNKAC
|
7.0 | IC50 | 4 | — | |
FNVQWFPDIYQCSF
|
7.0 | pIC50 | 8 | Yes | |
HIQIMBYLAJXNOK
|
7.0 | pIC50 | 3 | Yes | |
JEESDCKVMQTTMP
|
7.0 | Ki | 3 | — | |
OSVUGUHRKMMBSE
|
7.0 | Kd | 170 | — | |
SQYOZDZCDXQDRZ
|
7.0 | pIC50 | 3 | Yes | |
FHFXXELCOMBVAO
|
7.0 | pIC50 | 2 | Yes | |
KJAGZTFLBMDQQT
|
7.0 | pIC50 | 3 | Yes | |
CEUGFEWLHGCQEO
|
6.9 | pIC50 | 3 | Yes | |
ZATGFXTWDKIEKC
|
6.9 | pIC50 | 8 | Yes | |
CSFNNUIZTRGKSQ
|
6.9 | pIC50 | 3 | Yes | |
FGVBXWYMYMNXGE
|
6.9 | pIC50 | 4 | Yes | |
LQZVTJLMRRUWTJ
|
6.9 | pIC50 | 5 | Yes | |
MENIKIFJGYYVNI
|
6.9 | pIC50 | 5 | Yes | |
NSQXHPWPAPWSLN
|
6.9 | pIC50 | 3 | Yes | |
RETUSTLIJKZUGV
|
6.9 | pIC50 | 5 | Yes | |
JDNWHCLQTRJTAJ
|
6.9 | pIC50 | 6 | Yes | |
MZDKLVOWGIOKTN
|
6.9 | Kd | 80 | — | |
KDKUVYLMPJIGKA
|
6.8 | Kd | 91 | Yes | |
OAIDOYYRSBXKJG
|
6.8 | pIC50 | 3 | Yes | |
VQRJYECHVOWPDV
|
6.8 | pIC50 | 6 | Yes | |
DCYHJVFMNYSPNT
|
6.8 | IC50 | 9 | — | |
SCRSXZZGUOEUBI
|
6.8 | pIC50 | 4 | Yes | |
DPCPNRYPXUUJCP
|
6.8 | Ki | 4 | — | |
VBNPWXWJZJNXEY
|
6.8 | pIC50 | 18 | Yes | |
CNWZWPQCJCOBHA
|
6.8 | pIC50 | 3 | Yes | |
FHSKCOBLBQSSQE
|
6.8 | pIC50 | 3 | Yes | |
HBNGNYDOGUNIOV
|
6.8 | pIC50 | 2 | Yes | |
WVZWFOGYDXWKPT
|
6.8 | pIC50 | 5 | Yes | |
GJYVLTPTDBQQCY
|
6.8 | IC50 | 7 | — | |
IJXKSFMGCXZEEN
|
6.8 | pIC50 | 3 | Yes | |
ZIJIMHMKDXTURQ
|
6.8 | pIC50 | 6 | Yes | |
CJIAUJUVHMAHQC
|
6.7 | Ki | 4 | — | |
DRKOUHSEDVEHEG
|
6.7 | pIC50 | 3 | Yes | |
FFNIWOOLZGAOAB
|
6.7 | pIC50 | 8 | Yes | |
NTOMZGNNDKIPEH
|
6.7 | Ki | 4 | — | |
RIBFZRWGJCKRQH
|
6.7 | pIC50 | 3 | Yes | |
VNBRGSXVFBYQNN
|
6.7 | pIC50 | 22 | Yes | |
DKZYXHCYPUVGAF
|
6.7 | Kd | 112 | — | |
IAYJLHOAEWIYAY
|
6.7 | pIC50 | 4 | Yes | |
QLPKEICBTKFRKM
|
6.7 | pIC50 | 4 | Yes | |
HOHHMYNNRAVKQB
|
6.7 | pIC50 | 3 | Yes | |
YIHZVWLMRQCELC
|
6.7 | pIC50 | 3 | Yes | |
JIJYWPGTRDMEFZ
|
6.7 | pIC50 | 5 | Yes |