Target Details
| UniProt AC | O75716 |
|---|---|
| Gene Symbol | STK16 |
| Protein Name | Serine/threonine-protein kinase 16 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 456
- Clinical molecules 402
- Avg pChEMBL 7.28
Active Molecules (456)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VIHXUAKPZPXVSW
|
7.2 | pIC50 | 6 | Yes | |
BTQCPHBDUJMLMF
|
7.2 | pIC50 | 2 | Yes | |
VTKXOUFYFLRSDX
|
7.2 | pIC50 | 3 | Yes | |
CBLIPXTZSVBWET
|
7.2 | pIC50 | 3 | Yes | |
RBZINWUMPZNWCZ
|
7.2 | pIC50 | 4 | Yes | |
IZZAJZCFAZXNDC
|
7.2 | pIC50 | 6 | Yes | |
MOQBNQNUPNPLCH
|
7.2 | pIC50 | 7 | Yes | |
NACVPONJWZPHAP
|
7.2 | pIC50 | 5 | Yes | |
NYHVIVWBHLTODF
|
7.2 | pIC50 | 3 | Yes | |
XIZHRWKYFLKHBC
|
7.2 | pIC50 | 4 | Yes | |
PCTRICLZSMFSET
|
7.2 | pIC50 | 4 | Yes | |
WYLTWMHCCIFULE
|
7.2 | pIC50 | 3 | Yes | |
HEUIHAJXEGXNNB
|
7.2 | pIC50 | 2 | Yes | |
LMSNQXFIZAHXQB
|
7.2 | pIC50 | 3 | Yes | |
RGCULYFIEIGHSJ
|
7.2 | pIC50 | 2 | Yes | |
UNYZXVQYBXGDJS
|
7.2 | pIC50 | 2 | Yes | |
WMBJPWPAQLGSFL
|
7.2 | pIC50 | 6 | Yes | |
XKZQZMSAWVDRSP
|
7.2 | pIC50 | 39 | Yes | |
QRFIOQPCVMNZPT
|
7.2 | pIC50 | 3 | Yes | |
LEFKZSWCBZBDLU
|
7.2 | pIC50 | 5 | Yes | |
RBJQAHIBEYFAAG
|
7.2 | pIC50 | 3 | Yes | |
WVYZESHCWKLDBS
|
7.1 | pIC50 | 5 | Yes | |
JXKDTYDBDDKIPY
|
7.1 | pIC50 | 5 | Yes | |
SENOTLIGBLGKGP
|
7.1 | Ki | 3 | — | |
SRNHAKVSFVSSPN
|
7.1 | pIC50 | 8 | Yes | |
JNCRJZQZLMYLLM
|
7.1 | pIC50 | 3 | Yes | |
CEAQTTJXUPADGI
|
7.1 | pIC50 | 3 | Yes | |
CVMUHXWSBHMVGZ
|
7.1 | pIC50 | 6 | Yes | |
OEZHSZIDGUKBRK
|
7.1 | IC50 | 10 | — | |
ZFOPWBXSJXQVFA
|
7.1 | pIC50 | 3 | Yes | |
BBTDOQATPTVBOJ
|
7.1 | pIC50 | 3 | Yes | |
RDIZFHYTFVBBCX
|
7.1 | pIC50 | 2 | Yes | |
XQFHODAQACCOEF
|
7.1 | pIC50 | 3 | Yes | |
BGNRYQCGVJJPRI
|
7.1 | pIC50 | 3 | Yes | |
LEJNMWZPQMLOST
|
7.1 | pIC50 | 3 | Yes | |
PIQNNSKBFMKWGB
|
7.1 | pIC50 | 4 | Yes | |
RHDBNLYQAOUIAE
|
7.1 | pIC50 | 2 | Yes | |
YSMDVXCUNQWGNN
|
7.1 | Ki | 4 | — | |
ARQPPPCSTGSCQR
|
7.1 | pIC50 | 3 | Yes | |
RDROKTFULACVDQ
|
7.1 | IC50 | 8 | — | |
DCKMTGBFLNPJPS
|
7.0 | pIC50 | 4 | Yes | |
WZTHBTBWYVSGPF
|
7.0 | pIC50 | 4 | Yes | |
BOWWSMXUIIXBOU
|
7.0 | pIC50 | 3 | Yes | |
NQHMMDRPRXVCLT
|
7.0 | pIC50 | 8 | Yes | |
USXZHEGWWNBLBI
|
7.0 | Ki | 4 | — | |
HFSFBCFFSSYGFK
|
7.0 | pIC50 | 3 | Yes | |
KALSMXLQRKFVPO
|
7.0 | pIC50 | 3 | Yes | |
ZCCPLJOKGAACRT
|
7.0 | Kd | 599 | — | |
GAROAAIHALTJIR
|
7.0 | pIC50 | 3 | Yes | |
UVGSPPQDSXBTJW
|
7.0 | pIC50 | 2 | Yes |