Target Details
| UniProt AC | O75716 |
|---|---|
| Gene Symbol | STK16 |
| Protein Name | Serine/threonine-protein kinase 16 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 456
- Clinical molecules 402
- Avg pChEMBL 7.28
Active Molecules (456)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WOHBHEXSHHPQIV
|
9.4 | pIC50 | 8 | Yes | |
ZBNZXTGUTAYRHI
|
9.1 | pIC50 | 102 | Yes | |
AHFWDQSNXFITEU
|
9.0 | pIC50 | 4 | Yes | |
ATUGFOWGVANOHQ
|
9.0 | pIC50 | 4 | Yes | |
AYNBVKYDBZJRNM
|
9.0 | pIC50 | 2 | Yes | |
FNBGPMNXEGPANM
|
9.0 | pIC50 | 2 | Yes | |
GBJVVSCPOBPEIT
|
9.0 | pIC50 | 13 | Yes | |
GUKNWLMFOBWSRH
|
9.0 | pIC50 | 2 | Yes | |
HHFBDROWDBDFBR
|
9.0 | pIC50 | 40 | Yes | |
IBQHDBZMXPNKAU
|
9.0 | pIC50 | 2 | Yes | |
OTACRQCAOBRLAZ
|
9.0 | pIC50 | 8 | Yes | |
QYZOGCMHVIGURT
|
9.0 | pIC50 | 26 | Yes | |
SUIPNNKRHBDYHW
|
9.0 | pIC50 | 2 | Yes | |
XLXSRNTZHMLTMP
|
9.0 | pIC50 | 3 | Yes | |
ZLHFILGSQDJULK
|
9.0 | pIC50 | 37 | Yes | |
ZLLVQOSTXBHAIP
|
9.0 | pIC50 | 3 | Yes | |
VMAAFUOXTWPYRN
|
9.0 | pIC50 | 9 | Yes | |
XHHRGYCOEVNAKV
|
8.9 | pIC50 | 6 | Yes | |
XAQZJRAEQPCWMI
|
8.9 | pIC50 | 3 | Yes | |
MDHHYPFBVYJHPN
|
8.8 | pIC50 | 6 | Yes | |
CGLNKCUZVMEOBR
|
8.8 | pIC50 | 3 | Yes | |
FUIHJVJXGTVUJU
|
8.8 | pIC50 | 3 | Yes | |
LCQYMDMUCJFFKN
|
8.8 | pIC50 | 5 | Yes | |
MOSKATHMXWSZTQ
|
8.8 | pIC50 | 16 | Yes | |
USFRNJSCBVCBFY
|
8.8 | pIC50 | 4 | Yes | |
ANTUVUVMQSIJBS
|
8.8 | pIC50 | 3 | Yes | |
NHHQJBCNYHBUSI
|
8.8 | Kd | 220 | — | |
DYAYBUDFGBTDNI
|
8.7 | pIC50 | 2 | Yes | |
JLBXEVHWZFQSBL
|
8.7 | pIC50 | 3 | Yes | |
RHGZQGXELRMGES
|
8.7 | pIC50 | 8 | Yes | |
XUAORJVHYWCADO
|
8.7 | pIC50 | 5 | Yes | |
LEWVUPUKJSFGLR
|
8.6 | pIC50 | 3 | Yes | |
ZUOHNZIRNKHHJE
|
8.6 | pIC50 | 3 | Yes | |
HOPYTUITHBXQSC
|
8.6 | pIC50 | 5 | Yes | |
DCQUEYKYABNNDA
|
8.5 | pIC50 | 5 | Yes | |
FLYNZEXUURBXAW
|
8.5 | pIC50 | 6 | Yes | |
KJMALBRUCRDMTE
|
8.5 | pIC50 | 6 | Yes | |
LNGVCHKMQJKHDR
|
8.5 | pIC50 | 6 | Yes | |
LYDTZBUSUCDSRL
|
8.5 | pIC50 | 3 | Yes | |
PEPCSEJJADXCRB
|
8.5 | pIC50 | 4 | Yes | |
PGYJINWZLJSDIT
|
8.5 | pIC50 | 2 | Yes | |
PIRRYRRDDTYFPP
|
8.5 | pIC50 | 4 | Yes | |
AKSIZPIFQAYJGF
|
8.5 | pIC50 | 4 | Yes | |
CMEKRUHUVGTVLK
|
8.5 | pIC50 | 6 | Yes | |
LOLPPWBBNUVNQZ
|
8.5 | pIC50 | 97 | Yes | |
BRVRJAZHVITNIF
|
8.4 | pIC50 | 3 | Yes | |
AGHMFEHJWZVACU
|
8.4 | pIC50 | 3 | Yes | |
GBXVVXZXFOFHSU
|
8.4 | pIC50 | 3 | Yes | |
COBLQYUYOHSZOW
|
8.4 | pIC50 | 2 | Yes | |
DFAKFCGQJSYCEP
|
8.4 | pIC50 | 2 | Yes |