Target Details
| UniProt AC | O75676 |
|---|---|
| Gene Symbol | RPS6KA4 |
| Protein Name | Ribosomal protein S6 kinase alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 60
- Clinical molecules 15
- Avg pChEMBL 6.93
KEGG Pathways (2)
Active Molecules (60)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVKVSKQNYIHXPX
|
6.2 | Ki | 7 | — | |
ZHJGWYRLJUCMRT
|
6.1 | Kd | 18 | — | |
KBGCWMXCIHNWOI
|
6.1 | IC50 | 2 | — | |
XOVPCPRZRHQFBI
|
6.1 | Ki | 15 | — | |
PROGKLMIRQVLRO
|
6.1 | IC50 | 12 | — | |
IAYGCINLNONXHY
|
6.1 | Kd | 50 | — | |
AZTMYWWWILJAKW
|
6.0 | Ki | 16 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |