Target Details
| UniProt AC | O75608 |
|---|---|
| Gene Symbol | LYPLA1 |
| Protein Name | Acyl-protein thioesterase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02230 (Abhydrolase_2) |
Summary
- Multi-target molecules 10
- Clinical molecules 0
- Avg pChEMBL 7.96
KEGG Pathways (2)
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
9.3 | Kd | 1075 | — | |
HVJGVPUJTPBPAM
|
8.6 | IC50 | 2 | — | |
NHXPDCZIJAVTAO
|
8.6 | IC50 | 2 | — | |
OAQBMRDGOXAQTK
|
8.4 | IC50 | 2 | — | |
ASVWFAVGLYUDFD
|
8.3 | IC50 | 3 | — | |
BBNSKPZTKKCLDP
|
8.2 | IC50 | 2 | — | |
SUOZFKPRCIPXMF
|
8.0 | IC50 | 2 | — | |
LPTMHNPBMQCQPG
|
7.8 | IC50 | 2 | — | |
OXKNHBBDOIMFFQ
|
6.5 | Ki | 2 | — | |
DTCLGBKBZSVSLS
|
6.0 | Ki | 2 | — |