Target Details
| UniProt AC | O75582 |
|---|---|
| Gene Symbol | RPS6KA5 |
| Protein Name | Ribosomal protein S6 kinase alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 157
- Clinical molecules 17
- Avg pChEMBL 6.98
KEGG Pathways (9)
Active Molecules (157)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RFVBRKXQYUDGIO
|
6.6 | Ki | 23 | — | |
XQVVPGYIWAGRNI
|
6.6 | Kd | 34 | — | |
DKZYXHCYPUVGAF
|
6.5 | Kd | 112 | — | |
OWRXHGAFWZFFCW
|
6.5 | Ki | 113 | — | |
PUPCRRRSBUYJAD
|
6.5 | Ki | 44 | Yes | |
SBFPHSVZEXSHTL
|
6.5 | Ki | 62 | — | |
SPMHGQZFMNZCBV
|
6.5 | Ki | 30 | Yes | |
SYSUZXPGQXEWCZ
|
6.5 | Ki | 10 | — | |
XMFUGSRATNLPRM
|
6.5 | Ki | 19 | — | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
AXRCEOKUDYDWLF
|
6.4 | Kd | 31 | — | |
DZSUJUOJJJCWGG
|
6.4 | Ki | 55 | Yes | |
MHCPAORAYMTGCZ
|
6.4 | Ki | 37 | — | |
QEWSTOOMTBAUAG
|
6.4 | Ki | 17 | — | |
QKPLUKMJEKRAJD
|
6.4 | Ki | 30 | Yes | |
WINHZLLDWRZWRT
|
6.4 | Ki | 66 | — | |
GXJSLIOOPZRPEV
|
6.3 | Ki | 34 | — | |
JIFGOPCFXJIPNK
|
6.3 | Ki | 5 | — | |
PAIFYAZSILXLBO
|
6.3 | Ki | 26 | — | |
RWEHAHIEUDLKGT
|
6.3 | Ki | 33 | — | |
TVEREFRWBLRPPJ
|
6.3 | Ki | 15 | — | |
VNGYQBMDQMDALH
|
6.3 | Ki | 25 | — | |
XJSFDMGICAWQFS
|
6.3 | Ki | 60 | — | |
XOVPCPRZRHQFBI
|
6.3 | Ki | 15 | — | |
XSDJOIOVIMPMHD
|
6.3 | Ki | 44 | — | |
ZVYLAQPDMUKXOT
|
6.3 | IC50 | 5 | — | |
DBXGGXLBTWZXBB
|
6.2 | Ki | 39 | — | |
DJRPFIWIDKXORZ
|
6.2 | Ki | 9 | — | |
DWTNLZZEPSCAIH
|
6.2 | Ki | 25 | — | |
IYOZTVGMEWJPKR
|
6.2 | Ki | 10 | — | |
LKUJDAHYLPICSE
|
6.2 | Ki | 24 | — | |
LRZYYIZFBXFSJB
|
6.2 | Ki | 69 | — | |
MPVGZUGXCQEXTM
|
6.2 | Ki | 61 | Yes | |
PTVPBWWDGZSEAF
|
6.2 | Ki | 63 | — | |
RIUZPIBUSOHUKF
|
6.2 | Ki | 23 | — | |
XIOOJUQFJYPVLA
|
6.2 | Ki | 17 | — | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
ODPGGGTTYSGTGO
|
6.1 | Kd | 153 | — | |
DJUSDFVEBBYFFL
|
6.1 | Ki | 27 | — | |
AGYRJOAGMDIFKL
|
6.1 | Ki | 17 | — | |
GCYXEGSPUDSZJY
|
6.1 | Ki | 82 | — | |
VKBFHTIUXUCYRQ
|
6.1 | Ki | 66 | — | |
PROGKLMIRQVLRO
|
6.1 | IC50 | 12 | — | |
DKXHSOUZPMHNIZ
|
6.0 | Ki | 51 | Yes | |
DYSRECIVMDGUQU
|
6.0 | Ki | 29 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JZTOUVBEZONDKA
|
6.0 | Ki | 80 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MDJCUXFFMNEBHG
|
6.0 | Ki | 13 | — |