Target Details
| UniProt AC | O75582 |
|---|---|
| Gene Symbol | RPS6KA5 |
| Protein Name | Ribosomal protein S6 kinase alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 157
- Clinical molecules 17
- Avg pChEMBL 6.98
KEGG Pathways (9)
Active Molecules (157)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SFPWNTQWFFNJIH
|
7.3 | Ki | 48 | — | |
VXYDJXMHISGSDA
|
7.3 | Ki | 59 | — | |
YOBIWCLAYQWPPW
|
7.2 | IC50 | 23 | — | |
BHSOPYVVEZFHDB
|
7.1 | Ki | 25 | Yes | |
CFIBXVQLBVNOHW
|
7.1 | Ki | 64 | — | |
DKSNLQYRZJKYOC
|
7.1 | Ki | 51 | — | |
HRZOUBQYVUXBNS
|
7.1 | Ki | 38 | — | |
OHPRWVPOPFGLJG
|
7.1 | Ki | 19 | — | |
UMTWTCVTRDYHQQ
|
7.1 | Ki | 56 | — | |
ZRQXCQXWTLVASO
|
7.1 | Ki | 36 | — | |
BBJXVAVUGRNQFP
|
7.1 | IC50 | 5 | — | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
HIUHVDROHDSKTC
|
7.0 | Ki | 20 | — | |
BPNUQXPIQBZCMR
|
7.0 | Ki | 60 | — | |
FDBPGAHVEGEARY
|
7.0 | Ki | 19 | — | |
MVJMMLFMPWITEJ
|
7.0 | Ki | 110 | — | |
YGEACCLUBSGMMJ
|
7.0 | Ki | 16 | — | |
ZKZXNDJNWUTGDK
|
6.9 | IC50 | 9 | — | |
HNXJWWRRSGDVIW
|
6.9 | Ki | 13 | — | |
MQRDVGBWWVWMEN
|
6.9 | Ki | 47 | — | |
OWDRQHVEJIYVOI
|
6.9 | Ki | 47 | — | |
XYZNKCSDQRKAFR
|
6.9 | Ki | 53 | — | |
HCRQPXYLXXLKPT
|
6.8 | IC50 | 5 | — | |
HFNKQEVNSGCOJV
|
6.8 | Kd | 65 | — | |
CTNPALGJUAXMMC
|
6.8 | Kd | 151 | — | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
HXDDWVMJYDULAZ
|
6.8 | Ki | 13 | — | |
KGPGFQWBCSZGEL
|
6.8 | Kd | 59 | Yes | |
SGHXFHRRWFLILP
|
6.8 | Ki | 29 | — | |
UPPGGRZNGRFDAU
|
6.8 | Ki | 21 | — | |
UTFXYGYVDDLJER
|
6.8 | Ki | 36 | — | |
SXRCGQAHDJRHJC
|
6.8 | IC50 | 4 | — | |
CLRFYTGANQZOBS
|
6.7 | Ki | 41 | — | |
GLMWKEAUVZDGKE
|
6.7 | Ki | 23 | — | |
HKZKELVPGXJIMW
|
6.7 | Ki | 41 | — | |
KBGCWMXCIHNWOI
|
6.7 | IC50 | 2 | — | |
MADCXGNPDBWPLM
|
6.7 | Ki | 25 | — | |
ULHGAQSVFPOUDY
|
6.7 | Ki | 43 | — | |
XZXHXSATPCNXJR
|
6.7 | Kd | 165 | Yes | |
YPJJSXBVVGPFHA
|
6.7 | Ki | 18 | — | |
BMGQWWVMWDBQGC
|
6.6 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.6 | Kd | 91 | Yes | |
ACNCCUVYXQGPKZ
|
6.6 | Ki | 31 | — | |
GMYYMEOGFRKSFS
|
6.6 | Ki | 29 | — | |
JSKUWFIZUALZLX
|
6.6 | Ki | 33 | — | |
LCGSWTFWYNYUKS
|
6.6 | Ki | 26 | — | |
MCCCQFAOMZMZKE
|
6.6 | Ki | 52 | — | |
OEEGUWWPGAZRIJ
|
6.6 | Ki | 21 | — | |
OLVBAUVSICCWEJ
|
6.6 | Ki | 39 | — | |
OSVUGUHRKMMBSE
|
6.6 | Kd | 170 | — |