Target Details
| UniProt AC | O75582 |
|---|---|
| Gene Symbol | RPS6KA5 |
| Protein Name | Ribosomal protein S6 kinase alpha-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 157
- Clinical molecules 17
- Avg pChEMBL 6.98
KEGG Pathways (9)
Active Molecules (157)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MBCJUIJWPYUEBX
|
9.3 | IC50 | 7 | — | |
YWTBGJGMTBHQTM
|
9.1 | Ki | 65 | — | |
FIFFDYNJQGROBO
|
9.0 | IC50 | 5 | — | |
CHTMRWQLNNRRFJ
|
8.9 | Ki | 70 | — | |
FCCMYBKAZCDQGX
|
8.8 | IC50 | 2 | — | |
PHWHNHYZZNJPLB
|
8.5 | IC50 | 3 | — | |
UGHABJRZQKZAHP
|
8.5 | IC50 | 6 | — | |
XLYVQVWMTOLDNL
|
8.4 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
8.4 | IC50 | 21 | — | |
NJPWCTYVEJIQBM
|
8.3 | Ki | 72 | — | |
NRGYZNJPCGRCLV
|
8.3 | Ki | 52 | — | |
WVWKMLRXXWPJFD
|
8.3 | Kd | 3 | — | |
SAZVRXTVWZAHBI
|
8.2 | IC50 | 4 | — | |
FYXRSVDHGLUMHB
|
8.2 | IC50 | 8 | — | |
MHGPJIHGGLSWFD
|
8.1 | IC50 | 8 | — | |
DSXXEELGXBCYNQ
|
8.1 | IC50 | 28 | Yes | |
MLGGUGPIWDHBAI
|
8.1 | IC50 | 10 | — | |
MLGGUGPIWDHBAI
|
8.1 | Ki | 33 | — | |
LXPVLMCYPWKNBD
|
8.0 | IC50 | 2 | — | |
IEQAHFTVGLZUBI
|
8.0 | IC50 | 8 | — | |
GRMVBDUZCLNCGD
|
8.0 | IC50 | 3 | — | |
IIRWNGPLJQXWFJ
|
7.9 | IC50 | 21 | — | |
PABLVBARXHFRFL
|
7.9 | Kd | 5 | — | |
AFZXKZNWMHCMPD
|
7.9 | IC50 | 2 | — | |
LXUZPJDXRCSLIZ
|
7.9 | IC50 | 2 | — | |
PHWHNHYZZNJPLB
|
7.8 | IC50 | 6 | Yes | |
RIIYKHQJSKRYKG
|
7.8 | IC50 | 3 | — | |
NEWAULHLLUCDPD
|
7.8 | Ki | 27 | — | |
XFWUTMHVDGPWLH
|
7.8 | Ki | 75 | — | |
AOBLBPWPSKBHSI
|
7.7 | Ki | 55 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 408 | — | |
JRVSFZKYQCETAH
|
7.7 | Ki | 19 | — | |
BGZVXNSBCSLMND
|
7.7 | IC50 | 5 | — | |
BSFNGHCTZDCQBF
|
7.6 | Ki | 93 | — | |
VGNKOJURPOHWJF
|
7.6 | Ki | 21 | — | |
WINHZLLDWRZWRT
|
7.5 | Kd | 201 | Yes | |
RSFBRAHCHZGZPB
|
7.5 | IC50 | 8 | — | |
GLDSKRNGVVYJAB
|
7.5 | Kd | 16 | — | |
SGZZQKMOFHIDKW
|
7.5 | Kd | 13 | — | |
LGHBDVLAHHANMX
|
7.5 | Ki | 53 | — | |
ORUUEFDGYYTXAF
|
7.5 | Ki | 26 | — | |
SEVCBWKJSOLMNQ
|
7.5 | Ki | 38 | — | |
GSXRCPJTNIGKSZ
|
7.4 | Ki | 43 | — | |
XAHJIRNRDAKTEF
|
7.4 | Ki | 18 | — | |
HKSZLNNOFSGOKW
|
7.4 | Kd | 213 | — | |
OZFFKOSQNBBYCA
|
7.4 | IC50 | 12 | — | |
DWZCDSLYZDTWQH
|
7.3 | IC50 | 5 | — | |
CUAJADFGIOFJQT
|
7.3 | IC50 | 3 | — | |
YOVNFNXUCOWYSG
|
7.3 | IC50 | 33 | Yes | |
NPLQZQGAZAUUTB
|
7.3 | Ki | 9 | — |