Target Details
| UniProt AC | O75417 |
|---|---|
| Gene Symbol | POLQ |
| Protein Name | DNA polymerase theta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00270 (DEAD) PF00476 (DNA_pol_A) PF25453 (DUF7898) PF00271 (Helicase_C) PF20470 (HTH_61) PF21099 (POLQ_helical) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 7.19
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PBBZMQSTYBBLDS
|
7.2 | IC50 | 2 | — | |
BWTOWBOMDHKCDB
|
7.2 | IC50 | 7 | — | |
UTWLDWAFEKZNCC
|
7.1 | IC50 | 2 | — |