Target Details
| UniProt AC | O75385 |
|---|---|
| Gene Symbol | ULK1 |
| Protein Name | Serine/threonine-protein kinase ULK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12063 (ATG1-like_MIT1) PF21127 (ATG1-like_MIT2) PF00069 (Pkinase) |
Summary
- Multi-target molecules 55
- Clinical molecules 5
- Avg pChEMBL 7.1
KEGG Pathways (10)
Active Molecules (55)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KTEIFNKAUNYNJU
|
6.0 | Kd | 114 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
UIARLYUEJFELEN
|
6.0 | Kd | 289 | Yes |