Target Details
| UniProt AC | O75385 |
|---|---|
| Gene Symbol | ULK1 |
| Protein Name | Serine/threonine-protein kinase ULK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12063 (ATG1-like_MIT1) PF21127 (ATG1-like_MIT2) PF00069 (Pkinase) |
Summary
- Multi-target molecules 55
- Clinical molecules 5
- Avg pChEMBL 7.1
KEGG Pathways (10)
Active Molecules (55)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
9.1 | Kd | 231 | Yes | |
KYPQUQARPVLCEI
|
8.8 | IC50 | 2 | — | |
QFSIUHFQOJVPBQ
|
8.8 | IC50 | 2 | — | |
KKISLZKMBSCLSS
|
8.5 | IC50 | 2 | — | |
UEZRAYLQPKCVRW
|
8.5 | IC50 | 2 | — | |
DLCOOKRUECVLCI
|
8.1 | IC50 | 3 | — | |
GVNUZZFMGGXPMN
|
8.1 | IC50 | 2 | — | |
PFZRXJIYAFANHP
|
8.1 | IC50 | 4 | — | |
WEFRCKPVMWDRAK
|
8.1 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
NHHQJBCNYHBUSI
|
7.8 | Kd | 220 | — | |
WINHZLLDWRZWRT
|
7.6 | Kd | 201 | Yes | |
RYYNGWLOYLRZLK
|
7.5 | Kd | 45 | — | |
SSMPZXRXMBEUFU
|
7.5 | IC50 | 4 | — | |
XKTUKRBLWOHYIL
|
7.5 | IC50 | 4 | — | |
FIVNKJOGCQTGHE
|
7.3 | IC50 | 2 | — | |
LMPCYUMUDIOPBH
|
7.3 | IC50 | 2 | — | |
MGCUCAILCSYREM
|
7.3 | IC50 | 2 | — | |
UKBGBACORPRCGG
|
7.3 | IC50 | 17 | — | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
HTSMUTPVZNMYSW
|
7.3 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
7.3 | Kd | 137 | Yes | |
GWRHBTXTQFLVSP
|
7.2 | IC50 | 2 | — | |
BQROJYIEHOOQBY
|
7.2 | IC50 | 2 | — | |
AQFMGFCVDBEMQE
|
7.2 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
7.1 | Kd | 151 | — | |
VAVXGGRQQJZYBL
|
7.1 | IC50 | 8 | — | |
YSCYSYZEYWGLFD
|
7.0 | IC50 | 2 | — | |
ILNHHNVWAGBGGW
|
7.0 | IC50 | 2 | — | |
NEXGBSJERNQRSV
|
7.0 | IC50 | 3 | — | |
IAYGCINLNONXHY
|
6.9 | Kd | 50 | — | |
ZYLHCSSOEGIFAO
|
6.9 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
6.9 | Kd | 200 | — | |
RAXZSEGXMBWYQK
|
6.8 | Kd | 21 | — | |
BFSMGDJOXZAERB
|
6.7 | Kd | 33 | — | |
IVUGFMLRJOCGAS
|
6.7 | Kd | 9 | — | |
CLYZLUAUBTXCPL
|
6.6 | IC50 | 7 | — | |
JOOXLOJCABQBSG
|
6.6 | Kd | 139 | — | |
HFNKQEVNSGCOJV
|
6.5 | Kd | 65 | — | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
IGTBKTSITITXQX
|
6.5 | IC50 | 2 | — | |
JJEFZXFMIWYUFB
|
6.5 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
6.5 | Kd | 165 | Yes | |
MWKSRKSEWLRPBL
|
6.4 | Kd | 1075 | — | |
MZHPEELZCYWEHG
|
6.4 | IC50 | 6 | — | |
FVHKTXLAWSFSNK
|
6.4 | IC50 | 4 | — | |
XUZMWHLSFXCVMG
|
6.1 | Kd | 24 | — | |
DYNHJHQFHQTFTP
|
6.1 | Kd | 38 | — | |
HUXYBQXJVXOMKX
|
6.1 | Kd | 28 | — | |
HGCJKDOLUCMPFE
|
6.0 | IC50 | 5 | — |