Target Details
| UniProt AC | O75376 |
|---|---|
| Gene Symbol | NCOR1 |
| Protein Name | Nuclear receptor corepressor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15784 (GPS2_interact) PF00249 (Myb_DNA-binding) |
Summary
- Multi-target molecules 58
- Clinical molecules 7
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (58)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWSMVLJLEXXRHR
|
10.2 | IC50 | 5 | — | |
YNOXQYPNBSQQEI
|
10.1 | IC50 | 5 | — | |
OHRURASPPZQGQM
|
9.8 | Ki | 14 | — | |
UPCFDQLGZODPFB
|
9.8 | Ki | 10 | Yes | |
HCEDLZCUHOEHNH
|
9.8 | IC50 | 5 | — | |
RTKIYFITIVXBLE
|
9.3 | Ki | 17 | Yes | |
RBVSKBDEAXWXGR
|
9.2 | IC50 | 7 | — | |
NRXMHGVXTYHHEY
|
8.9 | IC50 | 5 | — | |
OEVNYXUGKVJBIX
|
8.7 | IC50 | 5 | — | |
DHDVNZCBVBNUML
|
8.5 | IC50 | 5 | — | |
DJJICDKYOCVBNI
|
8.5 | IC50 | 5 | — | |
WSTLKKSKCYMNAA
|
8.4 | IC50 | 7 | — | |
KRCXZGYVOZSCSF
|
8.0 | IC50 | 9 | Yes | |
SMTXKVURUPJKNQ
|
7.9 | IC50 | 5 | — | |
WAEXFXRVDQXREF
|
7.9 | IC50 | 20 | Yes | |
YPQXVNKTJNZZFB
|
7.9 | IC50 | 4 | — | |
HPNRVPHONJCSQC
|
7.9 | IC50 | 5 | — | |
HMTJEOJSDFUEKT
|
7.8 | IC50 | 4 | — | |
QKNOLJBQLJGNKI
|
7.8 | Ki | 8 | Yes | |
ULVBVRHTPUIWJF
|
7.8 | IC50 | 5 | — | |
FXCUYPUWZLTQGM
|
7.8 | IC50 | 4 | — | |
IOAQGGPWYTVPJM
|
7.7 | IC50 | 5 | — | |
HRNLUBSXIHFDHP
|
7.7 | IC50 | 7 | Yes | |
JMODMXNTOJTCLH
|
7.6 | IC50 | 4 | — | |
YPQXVNKTJNZZFB
|
7.6 | IC50 | 3 | — | |
DMXROUYLQHFRCS
|
7.6 | Ki | 7 | Yes | |
DMXROUYLQHFRCS
|
7.6 | Ki | 4 | — | |
ZOVGTEFLPRZPLH
|
7.5 | IC50 | 3 | — | |
DMKHBMNHLWJUQI
|
7.5 | IC50 | 6 | — | |
HCPJONOCDRERJJ
|
7.4 | IC50 | 4 | — | |
AMDUCWJBYRMCNV
|
7.4 | IC50 | 4 | — | |
UPTHKGNCOWCZQD
|
7.3 | IC50 | 4 | — | |
HCPJONOCDRERJJ
|
7.3 | IC50 | 4 | — | |
GMJBHVCHBXJWGH
|
7.2 | IC50 | 3 | — | |
JLIOMTJQMCMPRL
|
7.2 | IC50 | 3 | — | |
NTUCJWZWDDQYER
|
7.1 | IC50 | 7 | — | |
SMTXKVURUPJKNQ
|
7.1 | IC50 | 4 | — | |
PBZSSSTWPPXXEK
|
7.1 | IC50 | 3 | — | |
RVTQYDDCOIFTGY
|
7.0 | IC50 | 3 | — | |
LOSMQVNNNADUOB
|
7.0 | IC50 | 4 | — | |
YRUAJZFECDBHMT
|
7.0 | IC50 | 8 | — | |
KFRUOFXRWUHHPE
|
7.0 | IC50 | 3 | — | |
BMEYTXZHJHHKPN
|
6.9 | IC50 | 4 | — | |
OHHKIRZGQVDOQY
|
6.9 | IC50 | 4 | — | |
UTQMWCHHCIKOKP
|
6.8 | IC50 | 4 | — | |
HYGFVHOHMCNSIF
|
6.7 | IC50 | 4 | — | |
UKNPNNJYGOJZRO
|
6.6 | IC50 | 4 | — | |
WXHHICFWKXDFOW
|
6.6 | IC50 | 12 | — | |
LBLSLSOENGWIHL
|
6.6 | IC50 | 2 | — | |
AXAUXMXVFLCQQK
|
6.6 | IC50 | 2 | — |