Target Details
| UniProt AC | O75173 |
|---|---|
| Gene Symbol | ADAMTS4 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF00090 (TSP_1) |
Summary
- Multi-target molecules 239
- Clinical molecules 41
- Avg pChEMBL 7.43
Active Molecules (239)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODOUKZOJMQSYME
|
6.5 | IC50 | 2 | — | |
RQCXYESMODRPPY
|
6.5 | IC50 | 4 | Yes | |
WRNVCIFWXDWAQY
|
6.5 | IC50 | 2 | — | |
WECKJJDCDPVTTO
|
6.4 | IC50 | 3 | — | |
YPTZORUBNMNKDA
|
6.4 | IC50 | 2 | — | |
CCTJPVSDIZDFJW
|
6.4 | IC50 | 3 | Yes | |
DXEOUZOCKYSZQC
|
6.4 | IC50 | 2 | — | |
HKBXBBXQCDCNLR
|
6.4 | IC50 | 2 | — | |
KNOYHJOPRUTPSQ
|
6.4 | Ki | 7 | — | |
WFKAOUORBBLUOE
|
6.4 | IC50 | 2 | — | |
IYBHJPNFVKYDOX
|
6.4 | IC50 | 3 | — | |
YINSFKOGVSNIAY
|
6.3 | IC50 | 2 | — | |
AWLKOGZBGNQOBA
|
6.3 | IC50 | 5 | Yes | |
QOPRVQPJWCZITD
|
6.3 | IC50 | 2 | — | |
NITYDPDXAAFEIT
|
6.3 | IC50 | 20 | Yes | |
XZMNHVVTOKEKOE
|
6.3 | IC50 | 2 | — | |
IABWDXKLHPEEBX
|
6.3 | IC50 | 2 | — | |
OYJHJMVVIQMCQV
|
6.3 | IC50 | 2 | — | |
JPZUAZMIFKHSGZ
|
6.3 | IC50 | 2 | — | |
HECFJRXDSZZJLW
|
6.3 | IC50 | 3 | Yes | |
CRWSSUTUNYHTON
|
6.3 | IC50 | 2 | — | |
YJRJYIQWWPZSTM
|
6.2 | IC50 | 6 | — | |
VFHNZPCBNRDGLE
|
6.2 | IC50 | 2 | — | |
FGQTUBBIXYISNM
|
6.2 | IC50 | 4 | — | |
JRAYHZWPXHIVJI
|
6.2 | IC50 | 2 | — | |
UJRBIZNZOPPPEC
|
6.2 | IC50 | 2 | — | |
CNVJYZPKUZXAML
|
6.2 | IC50 | 4 | Yes | |
PPCHUKYNNDWTFT
|
6.2 | IC50 | 3 | — | |
RPVHARCGZZMFFN
|
6.2 | IC50 | 2 | — | |
ASVLCJFACSELPH
|
6.1 | IC50 | 2 | — | |
BSYDZRAGBLIBSI
|
6.1 | IC50 | 2 | — | |
HOSYCMQDQLQXLY
|
6.1 | IC50 | 2 | — | |
DJEDDHGTONHFQL
|
6.1 | IC50 | 2 | — | |
RIJMYCAFDDBRHW
|
6.1 | IC50 | 2 | — | |
YDMFQFGWICWKSM
|
6.1 | IC50 | 2 | — | |
WNKWHJMCHLXGLE
|
6.1 | IC50 | 2 | — | |
IMKDKHQDFFLOKK
|
6.0 | IC50 | 13 | Yes | |
IOBCRLWDQPOVFD
|
6.0 | IC50 | 2 | — | |
SRNVCZIFDUXAJE
|
6.0 | IC50 | 2 | — |