Target Details
| UniProt AC | O75173 |
|---|---|
| Gene Symbol | ADAMTS4 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF00090 (TSP_1) |
Summary
- Multi-target molecules 239
- Clinical molecules 41
- Avg pChEMBL 7.43
Active Molecules (239)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UUIVHPQOLWYKFC
|
7.1 | IC50 | 3 | — | |
XZQFSKBVCGYHFA
|
7.1 | IC50 | 3 | — | |
ZEMLAXHMFOILNW
|
7.1 | IC50 | 3 | — | |
CHTZMALPRVCUIK
|
7.1 | IC50 | 4 | — | |
ONWZTEISEVDFER
|
7.1 | IC50 | 2 | — | |
ZHXMXRVBOZWQPF
|
7.1 | IC50 | 5 | Yes | |
WZHCTLSXWLCZEU
|
7.1 | IC50 | 2 | — | |
LPGGJWIOKRQQAT
|
7.1 | IC50 | 2 | — | |
CYVZQRKPMGDNKM
|
7.0 | IC50 | 4 | Yes | |
BHHZCJUKKKCRHQ
|
7.0 | IC50 | 2 | — | |
CQARAIRTGMAYMZ
|
7.0 | Ki | 8 | — | |
JKTGELXOMXEKJI
|
7.0 | IC50 | 2 | Yes | |
CHUAOQGPMXWHAQ
|
7.0 | IC50 | 2 | — | |
CVZIHNYAZLXRRS
|
7.0 | IC50 | 10 | Yes | |
IBSGSCYXBWXQDW
|
7.0 | IC50 | 4 | Yes | |
JGTIIKHYSZFICL
|
7.0 | IC50 | 5 | Yes | |
MBFFAPVZPKHCKK
|
7.0 | IC50 | 2 | — | |
QDUBONLFDSIPOU
|
7.0 | IC50 | 2 | — | |
UWLVDBFIOGAENY
|
7.0 | IC50 | 2 | — | |
ZPCSCHFHONOZPV
|
7.0 | IC50 | 2 | — | |
GPHYVVDMOPSOAK
|
7.0 | IC50 | 2 | — | |
IKHZGIGQISAUFN
|
7.0 | IC50 | 2 | — | |
STVUCRKRBAWCPC
|
7.0 | IC50 | 4 | Yes | |
YGEZZRWSTUOZOA
|
7.0 | IC50 | 2 | — | |
KDDWLGBIYXTPJG
|
7.0 | Ki | 5 | — | |
ICYKNMGQZVFJRC
|
6.9 | IC50 | 2 | — | |
RAAOGGVTKNNZQU
|
6.9 | IC50 | 2 | — | |
USQGYAOLZCMMRG
|
6.9 | IC50 | 2 | — | |
WRNVCIFWXDWAQY
|
6.9 | IC50 | 2 | — | |
OFQBKLDPHHFEPJ
|
6.9 | IC50 | 2 | Yes | |
SPZLSWDAZSYJAK
|
6.8 | IC50 | 2 | — | |
FLTAYQGSMZKKCR
|
6.8 | IC50 | 2 | — | |
CMLVKUWQFZQPPS
|
6.8 | IC50 | 3 | — | |
OBXOKKGDFARJJV
|
6.8 | IC50 | 2 | — | |
ZGUHWFRFXRBHPL
|
6.8 | IC50 | 2 | — | |
CSFRMTJLCGWESV
|
6.8 | IC50 | 2 | — | |
OYVRPNKMOGLOSV
|
6.8 | IC50 | 2 | — | |
RVGJJKGKACPPHF
|
6.8 | IC50 | 2 | — | |
ZRAVABUPGXTUEH
|
6.8 | IC50 | 2 | — | |
AUSYXXOLFARXLL
|
6.7 | IC50 | 2 | — | |
FNCXJJHZBHAVJZ
|
6.7 | IC50 | 2 | — | |
IOOCYYNMZOYCGW
|
6.6 | IC50 | 2 | — | |
OJALZWLVBUFAQK
|
6.6 | IC50 | 4 | Yes | |
OYVHTQLDQCPMLV
|
6.6 | IC50 | 2 | — | |
MASAPOBQXDWROW
|
6.6 | IC50 | 2 | — | |
LJEOQKRAJXJUKV
|
6.6 | IC50 | 2 | — | |
ZMONONWLGUTMJN
|
6.6 | IC50 | 2 | — | |
ALDHNIAORPZUFG
|
6.5 | IC50 | 2 | — | |
VPPAFDVKUDHCGQ
|
6.5 | IC50 | 2 | — | |
IENKEAFTWAFNOL
|
6.5 | IC50 | 2 | — |