Target Details
| UniProt AC | O75173 |
|---|---|
| Gene Symbol | ADAMTS4 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF00090 (TSP_1) |
Summary
- Multi-target molecules 239
- Clinical molecules 41
- Avg pChEMBL 7.43
Active Molecules (239)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FFYZDEBNTHTQDB
|
7.4 | IC50 | 3 | — | |
HVVNIZVKUPEBRS
|
7.4 | IC50 | 3 | — | |
JSUBEBYUGKGELF
|
7.4 | IC50 | 3 | — | |
LTDJFOLMHATVKC
|
7.4 | IC50 | 3 | — | |
MDCDJAYEONMPDM
|
7.4 | IC50 | 3 | — | |
MSDBLKCNXKEOHU
|
7.4 | IC50 | 3 | — | |
RDAJPGITRGURGP
|
7.4 | IC50 | 3 | — | |
RDWFDWWQRNYJGA
|
7.4 | IC50 | 3 | — | |
RKELHXSYFGUUBO
|
7.4 | IC50 | 3 | — | |
VUBCFWBRGYOPKR
|
7.4 | IC50 | 3 | — | |
OTYJRWAMIOUIHN
|
7.4 | IC50 | 4 | Yes | |
RZYRWVVQRWYGNG
|
7.4 | IC50 | 2 | — | |
MXNKXPGDSQYTQD
|
7.4 | IC50 | 2 | — | |
HGVMZFIYNIXZLZ
|
7.4 | IC50 | 2 | — | |
HTKFMVXDGZGNNW
|
7.4 | IC50 | 2 | — | |
CTRAVVYZOOTOPH
|
7.4 | IC50 | 2 | — | |
ZMZUPFGBAXDKAM
|
7.4 | IC50 | 2 | — | |
MBFFAPVZPKHCKK
|
7.4 | IC50 | 2 | — | |
QMEYEEICXNLCJY
|
7.4 | IC50 | 2 | — | |
DYWJWAJWDDNBGQ
|
7.3 | IC50 | 2 | — | |
RVGJJKGKACPPHF
|
7.3 | IC50 | 2 | — | |
QMEYEEICXNLCJY
|
7.3 | IC50 | 2 | — | |
RVGJJKGKACPPHF
|
7.3 | IC50 | 2 | — | |
LBFZDWQGADLLKS
|
7.3 | IC50 | 2 | — | |
MNKVQIVVYRSCJP
|
7.3 | IC50 | 2 | — | |
RSWPLKVUMZDBKI
|
7.3 | IC50 | 2 | — | |
UOXSWFRPRZUDSH
|
7.3 | IC50 | 2 | — | |
XWNLDJDYIDRBJI
|
7.3 | IC50 | 2 | — | |
AABQMYBVWBDBKY
|
7.2 | IC50 | 2 | — | |
DHURRPCJMDEPTJ
|
7.2 | IC50 | 2 | — | |
GNBHJTYIJMLFLC
|
7.2 | Ki | 6 | — | |
NWJMYUBNMRZMDU
|
7.2 | IC50 | 2 | — | |
LYUGBLDGSRTMRP
|
7.2 | IC50 | 2 | — | |
RSWPLKVUMZDBKI
|
7.2 | IC50 | 2 | — | |
WRNVCIFWXDWAQY
|
7.2 | IC50 | 2 | — | |
VXDKQRWTOJFQKH
|
7.2 | IC50 | 3 | Yes | |
ZQBRQDVCSATBBO
|
7.2 | IC50 | 2 | — | |
LNIRXDCIYOBRPL
|
7.1 | IC50 | 3 | — | |
XVMVNUAGECGGNK
|
7.1 | IC50 | 2 | — | |
ABNKQEYPWPPOOQ
|
7.1 | IC50 | 3 | — | |
AVLVMNPMCNZRPM
|
7.1 | IC50 | 3 | — | |
CMCAGYNSFUQZEV
|
7.1 | IC50 | 2 | — | |
CWKIDLOBKBRJAS
|
7.1 | IC50 | 2 | — | |
DNPHOKZQIKLZJT
|
7.1 | IC50 | 2 | — | |
HBRVHODOXCBKHN
|
7.1 | IC50 | 3 | — | |
IHRJQBVRWWFMFZ
|
7.1 | IC50 | 3 | — | |
KQDWIZNOSHZMAC
|
7.1 | IC50 | 3 | — | |
MDCDJAYEONMPDM
|
7.1 | IC50 | 3 | — | |
NAZJMGDZKSUZPA
|
7.1 | IC50 | 3 | — | |
QJRMCRVDHSDQOQ
|
7.1 | IC50 | 3 | — |