Target Details
| UniProt AC | O75173 |
|---|---|
| Gene Symbol | ADAMTS4 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF00090 (TSP_1) |
Summary
- Multi-target molecules 239
- Clinical molecules 41
- Avg pChEMBL 7.43
Active Molecules (239)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WJULIBHPWZXMJA
|
8.1 | IC50 | 10 | Yes | |
DNZQEIOYACTIFD
|
8.1 | IC50 | 2 | — | |
PSAIRTKPKUWNNP
|
8.0 | IC50 | 2 | — | |
IIJIMCYNCLMHHL
|
8.0 | IC50 | 2 | — | |
MAQGKYQDMNIZTG
|
8.0 | IC50 | 2 | — | |
ZRQWUQCXSKEXGA
|
8.0 | Ki | 6 | — | |
DDRRRYMVRWYNKI
|
8.0 | IC50 | 2 | — | |
QWGZIDLVLODPRW
|
8.0 | IC50 | 2 | — | |
UKSOPPJLMFZIFG
|
8.0 | IC50 | 2 | — | |
GYAIYJXOPICREB
|
7.9 | IC50 | 2 | — | |
KDEHHSHGVKUYEZ
|
7.9 | IC50 | 3 | — | |
NPTUUUXCZCQNQS
|
7.9 | IC50 | 5 | — | |
OBQNFIXICFYDBT
|
7.9 | IC50 | 3 | — | |
UOXSWFRPRZUDSH
|
7.9 | IC50 | 2 | — | |
VJASAEQMGHZSFE
|
7.9 | IC50 | 2 | — | |
BEYBREWPWQEWSI
|
7.9 | IC50 | 3 | — | |
BTKROMQYNIJXLC
|
7.9 | IC50 | 2 | — | |
VJASAEQMGHZSFE
|
7.8 | IC50 | 2 | — | |
VXXYNKXMRXANKX
|
7.8 | IC50 | 2 | — | |
HRHIVHWFCGOVGL
|
7.8 | IC50 | 2 | — | |
KTSVBNSBXWVDTE
|
7.8 | IC50 | 3 | — | |
MAQGKYQDMNIZTG
|
7.8 | IC50 | 2 | — | |
IWRJDNKXMJBFEA
|
7.8 | IC50 | 2 | — | |
OACIIQIUQKQGAD
|
7.8 | IC50 | 2 | — | |
SFQHPECSYRCUKU
|
7.8 | IC50 | 2 | — | |
WIKRDIGSYVQGTH
|
7.8 | IC50 | 2 | — | |
QMEYEEICXNLCJY
|
7.7 | IC50 | 2 | — | |
RKYYWBHSYPIJKC
|
7.7 | IC50 | 4 | — | |
LHERXAOZMZIVQX
|
7.7 | IC50 | 2 | — | |
CAFLLFZUWQCIHM
|
7.7 | IC50 | 2 | — | |
MOWYZZPAPKVBEC
|
7.7 | IC50 | 2 | — | |
OUTUIYKUSHWASL
|
7.7 | IC50 | 2 | — | |
ZQBRQDVCSATBBO
|
7.7 | IC50 | 2 | — | |
BMAHWOMMEYMRNY
|
7.7 | IC50 | 2 | — | |
CSFRMTJLCGWESV
|
7.7 | IC50 | 2 | — | |
SZDCEHDWAAZEPH
|
7.7 | IC50 | 2 | — | |
RDRCRROFSMSFED
|
7.6 | IC50 | 2 | — | |
RDRCRROFSMSFED
|
7.6 | IC50 | 2 | — | |
JHWOJEJVRYYQFM
|
7.6 | IC50 | 2 | — | |
UOXSWFRPRZUDSH
|
7.6 | IC50 | 2 | — | |
FWVMIBWFTPZCBI
|
7.6 | IC50 | 2 | — | |
SZEOXTMGYZKQHV
|
7.6 | IC50 | 4 | — | |
ISHINUUQDKDNHQ
|
7.6 | IC50 | 2 | — | |
NXFDHNJDXVCAMS
|
7.6 | IC50 | 2 | — | |
OGDMRINQXHOSNB
|
7.5 | IC50 | 2 | — | |
FKHNOEWOJMNEPT
|
7.5 | IC50 | 2 | — | |
LHKXLEZLEFHFJV
|
7.5 | IC50 | 3 | — | |
GYSTVJYXBPSVIF
|
7.5 | Ki | 4 | — | |
BVFMJFRMGBKBIW
|
7.4 | IC50 | 3 | — | |
CVXZBZOHZGZICE
|
7.4 | IC50 | 3 | — |