Target Details
| UniProt AC | O75173 |
|---|---|
| Gene Symbol | ADAMTS4 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF00090 (TSP_1) |
Summary
- Multi-target molecules 239
- Clinical molecules 41
- Avg pChEMBL 7.43
Active Molecules (239)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXKRFERDVUXQLW
|
9.7 | IC50 | 6 | Yes | |
YAQNYFRHXMKRGE
|
9.6 | IC50 | 3 | Yes | |
UDTXDKDGZMYOBK
|
9.4 | IC50 | 5 | Yes | |
SOTNGZPOQMJOPI
|
9.4 | IC50 | 2 | — | |
AFXZHRNVMMQHOL
|
9.3 | IC50 | 4 | Yes | |
KFGJNQLPIZMSFB
|
9.3 | IC50 | 5 | Yes | |
NYJKRUFCTNREQN
|
9.3 | IC50 | 3 | Yes | |
AYZCFZMCYDMFMY
|
9.3 | IC50 | 4 | Yes | |
JGAIDLBSMBNOAG
|
9.3 | IC50 | 4 | Yes | |
BWHNAQMOABQLDB
|
9.2 | IC50 | 4 | Yes | |
UAGAABCJKYADIR
|
9.2 | IC50 | 3 | — | |
BGUXTVRZPYKBBN
|
9.0 | IC50 | 5 | Yes | |
LTVIJEFEZVFIST
|
9.0 | IC50 | 14 | Yes | |
GBGAKFWYCGVPHY
|
9.0 | IC50 | 7 | Yes | |
DWKKNTWUNOATQS
|
8.9 | IC50 | 2 | — | |
SIXCEPSXNLUZTE
|
8.9 | IC50 | 2 | — | |
BZUGNOPIQMYMFU
|
8.8 | IC50 | 2 | — | |
KLCHUAUMSZUJEX
|
8.8 | IC50 | 5 | Yes | |
NPTUUUXCZCQNQS
|
8.8 | IC50 | 4 | — | |
USZJYBQKSJDVGU
|
8.8 | IC50 | 2 | — | |
VKMTZVHITCDFFV
|
8.7 | IC50 | 2 | — | |
JHOUEQAOHDTLPY
|
8.7 | IC50 | 4 | — | |
XTJBTJMEXZEGIF
|
8.7 | IC50 | 6 | — | |
SVXOKXGEZUGFFS
|
8.7 | IC50 | 3 | Yes | |
VLNVWKDSFQRXHZ
|
8.6 | IC50 | 5 | Yes | |
JAPLGNWCNXCEJT
|
8.6 | IC50 | 5 | Yes | |
LDIAENRSEDNGCJ
|
8.5 | IC50 | 2 | — | |
NPWGFJCNOCYDSO
|
8.5 | IC50 | 2 | — | |
UACUZULRKJKTHE
|
8.5 | IC50 | 5 | Yes | |
YSYXAGMNRKARQB
|
8.5 | IC50 | 4 | Yes | |
CVBUIFHDZMEAIE
|
8.4 | IC50 | 2 | — | |
GRSFKJZRDUZQPW
|
8.4 | IC50 | 9 | Yes | |
LDDKAYGLGQWILO
|
8.4 | IC50 | 6 | — | |
PDBQNZHFRVAZBC
|
8.4 | IC50 | 2 | — | |
PKTAGMTUNRVAKO
|
8.4 | IC50 | 2 | — | |
YGTSAUDEZYDSGM
|
8.4 | IC50 | 2 | — | |
NYSZVCQWENKRKM
|
8.3 | IC50 | 5 | Yes | |
LBFZDWQGADLLKS
|
8.3 | IC50 | 2 | — | |
DVWZDEQXQWWQOU
|
8.2 | IC50 | 3 | — | |
VYEJHVQIVKCLHC
|
8.2 | IC50 | 4 | Yes | |
INOYENJSYPDBEC
|
8.2 | IC50 | 3 | — | |
SPAODDWHKVLWKW
|
8.2 | IC50 | 2 | — | |
CHUAOQGPMXWHAQ
|
8.2 | IC50 | 2 | — | |
FJEJHTFPLBTMLO
|
8.2 | IC50 | 4 | — | |
LDIAENRSEDNGCJ
|
8.2 | IC50 | 2 | — | |
MEGFCBVTRXVKDO
|
8.1 | IC50 | 6 | Yes | |
AONLPKICQLHFDZ
|
8.1 | IC50 | 2 | — | |
LBFZDWQGADLLKS
|
8.1 | IC50 | 2 | — | |
LBVBVIKJOWWVJX
|
8.1 | IC50 | 4 | — | |
VJASAEQMGHZSFE
|
8.1 | IC50 | 2 | — |