Target Details
| UniProt AC | O75164 |
|---|---|
| Gene Symbol | KDM4A |
| Protein Name | Lysine-specific demethylase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02373 (JmjC) PF02375 (JmjN) PF13831 (PHD_2) PF18104 (Tudor_2) PF13832 (zf-HC5HC2H_2) |
Summary
- Multi-target molecules 140
- Clinical molecules 0
- Avg pChEMBL 6.68
Active Molecules (140)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ONKWECDQZPASOC
|
6.3 | IC50 | 4 | — | |
QVSDPEWGBYKEDU
|
6.3 | IC50 | 4 | — | |
TYQVGBHPIVDCJP
|
6.3 | IC50 | 4 | — | |
VBYNYZPZKXJUEM
|
6.3 | IC50 | 3 | — | |
VJLABPNSGBCXOH
|
6.3 | IC50 | 2 | — | |
VTBZXRRFAQZNQE
|
6.3 | IC50 | 2 | — | |
WAPIESSEOAYVNJ
|
6.3 | IC50 | 5 | — | |
WEZPYYZPYXGXHK
|
6.3 | IC50 | 2 | — | |
WIFDYYDCPDNMJO
|
6.3 | IC50 | 2 | — | |
WJNMKYLJNLYALB
|
6.3 | IC50 | 4 | — | |
WTMJZFIQFSYVHA
|
6.3 | IC50 | 4 | — | |
YEIUTPICFPHMSZ
|
6.3 | IC50 | 4 | — | |
YMWREFXLGWZZOR
|
6.3 | IC50 | 5 | — | |
ZQNXWEZQRNBWCU
|
6.3 | IC50 | 5 | — | |
KWVQXVRPRJIRSJ
|
6.2 | IC50 | 4 | — | |
UAKCGLKAUUAKCL
|
6.2 | IC50 | 4 | — | |
XYBBSEAKIBCXQV
|
6.2 | IC50 | 4 | — | |
YFRHLEVQXDGTNW
|
6.2 | IC50 | 2 | — | |
IALMMJCSQDGXBB
|
6.2 | IC50 | 5 | — | |
ZTYRLXUTLYBVHH
|
6.2 | IC50 | 8 | — | |
FGIPAHGTFZFKQH
|
6.2 | IC50 | 4 | — | |
CLDDHWNJFOWJLH
|
6.2 | IC50 | 4 | — | |
MJIVRKPEXXHNJT
|
6.2 | IC50 | 9 | — | |
XIMIJJARGYSDBU
|
6.1 | IC50 | 4 | — | |
FWXNBMPVCHFMRX
|
6.1 | IC50 | 4 | — | |
ARDXICZNEUJDDE
|
6.1 | IC50 | 5 | — | |
SBOZGYUGKHFCFF
|
6.1 | IC50 | 3 | — | |
WXDMSMYTZQAHRC
|
6.1 | IC50 | 4 | — | |
INPKYGJHWGXUDF
|
6.1 | IC50 | 4 | — | |
NLGUSOLKPNWPKR
|
6.0 | IC50 | 4 | — | |
VHUXANZSWRXPQK
|
6.0 | IC50 | 4 | — | |
BJPPOTJAQZGVIA
|
6.0 | IC50 | 4 | — | |
IBSVWTKUXPGZFI
|
6.0 | IC50 | 3 | — | |
GGAYQPAKFUJHFR
|
6.0 | IC50 | 3 | — | |
IGXZIIVCDBVBSB
|
6.0 | IC50 | 2 | — | |
JQPYWFPJAZZKAV
|
6.0 | IC50 | 5 | — | |
RHPSPIUSPOTEGT
|
6.0 | IC50 | 2 | — | |
UDNZKYWBVTTWJF
|
6.0 | IC50 | 5 | — | |
WVEHUIVVPBXOJC
|
6.0 | IC50 | 5 | — | |
YYOBYQZCYKMCFA
|
6.0 | IC50 | 4 | — |