Target Details
| UniProt AC | O75164 |
|---|---|
| Gene Symbol | KDM4A |
| Protein Name | Lysine-specific demethylase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02373 (JmjC) PF02375 (JmjN) PF13831 (PHD_2) PF18104 (Tudor_2) PF13832 (zf-HC5HC2H_2) |
Summary
- Multi-target molecules 140
- Clinical molecules 0
- Avg pChEMBL 6.68
Active Molecules (140)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SQDIBEJSOSAPGF
|
6.9 | IC50 | 4 | — | |
RIVJXVMWOIAAEH
|
6.8 | IC50 | 4 | — | |
DDRYBCASNXOENV
|
6.8 | IC50 | 4 | — | |
JOPSCFKAECJOQR
|
6.8 | IC50 | 4 | — | |
XIVQRYFYMNIDET
|
6.8 | IC50 | 4 | — | |
YAWHCFISAFZXHF
|
6.8 | IC50 | 4 | — | |
AIEULFAFWDPGEJ
|
6.8 | IC50 | 4 | — | |
RZAREOJWVVYJGA
|
6.8 | IC50 | 4 | — | |
DUTYNXONGTVYED
|
6.8 | IC50 | 4 | — | |
RRZDZCQQAMZZMU
|
6.8 | IC50 | 4 | — | |
FBNVHXXPQQVJCQ
|
6.7 | IC50 | 4 | — | |
WMPDPRRYFWPZOM
|
6.7 | IC50 | 4 | — | |
OTYMAMBJVVRSCZ
|
6.7 | IC50 | 4 | — | |
FAOZNCYQMCTIBT
|
6.7 | IC50 | 6 | — | |
JGRPKOGHYBAVMW
|
6.7 | IC50 | 13 | — | |
VCITXXCATLNLDE
|
6.7 | IC50 | 4 | — | |
IHCQQEZDLLAALX
|
6.7 | IC50 | 4 | — | |
OFBASLHLTNSWOV
|
6.6 | IC50 | 4 | — | |
JKWOFYNSPFBQLX
|
6.6 | IC50 | 4 | — | |
KWCSIVPBRNLEDE
|
6.6 | IC50 | 2 | — | |
FSICLPHOMOJFQK
|
6.5 | IC50 | 4 | — | |
YHHFKWKMXWRVTJ
|
6.5 | IC50 | 7 | — | |
WAXTXDDUSDCZNA
|
6.5 | IC50 | 4 | — | |
RGGMVQDDHDCRDM
|
6.5 | IC50 | 9 | — | |
FKGOBFPQRRZPLE
|
6.5 | IC50 | 2 | — | |
TWKOGDIJEBKSKF
|
6.4 | IC50 | 4 | — | |
ZVDVVBQKFXBYJN
|
6.4 | IC50 | 4 | — | |
OZMKCTFOIBLWOO
|
6.4 | IC50 | 5 | — | |
QDNXWZJEOBANTA
|
6.4 | IC50 | 4 | — | |
VIUFHKFDQXQPJV
|
6.3 | IC50 | 4 | — | |
FYEQKMAVRYRMBL
|
6.3 | IC50 | 2 | — | |
LHYVGHNYNLLNOV
|
6.3 | IC50 | 4 | — | |
ABANEZXFVFHRMY
|
6.3 | IC50 | 2 | — | |
BNEDYWDXODJLAY
|
6.3 | IC50 | 5 | — | |
DYRCVDOEKTXODY
|
6.3 | IC50 | 2 | — | |
FEZIKLVLFANZBD
|
6.3 | IC50 | 4 | — | |
FNPHROKMXPECAD
|
6.3 | IC50 | 4 | — | |
FWSGIYDMJPQQGL
|
6.3 | IC50 | 4 | — | |
GMVQFVAPKMAASG
|
6.3 | IC50 | 2 | — | |
GUHGGLPTVJEQIO
|
6.3 | IC50 | 2 | — | |
HJHPUQDFLVHFFZ
|
6.3 | IC50 | 2 | — | |
HNQJHFKEFOZLKD
|
6.3 | IC50 | 2 | — | |
IDAVRDSVKYWQFM
|
6.3 | IC50 | 2 | — | |
IHQFUQDEYXBGQR
|
6.3 | IC50 | 2 | — | |
IKDUYJZLUXCOMP
|
6.3 | IC50 | 4 | — | |
JFUSDWYLUAUIKN
|
6.3 | IC50 | 5 | — | |
KPJOSXHPFIXXLA
|
6.3 | IC50 | 4 | — | |
LKBZHRSAENXIOI
|
6.3 | IC50 | 4 | — | |
LYECZDRRRZNARD
|
6.3 | IC50 | 2 | — | |
OMVZFTXWQQJIHI
|
6.3 | IC50 | 2 | — |