Target Details
| UniProt AC | O75164 |
|---|---|
| Gene Symbol | KDM4A |
| Protein Name | Lysine-specific demethylase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02373 (JmjC) PF02375 (JmjN) PF13831 (PHD_2) PF18104 (Tudor_2) PF13832 (zf-HC5HC2H_2) |
Summary
- Multi-target molecules 140
- Clinical molecules 0
- Avg pChEMBL 6.68
Active Molecules (140)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GFHQSNHGGSKSHQ
|
8.4 | IC50 | 2 | — | |
GFHQSNHGGSKSHQ
|
8.2 | IC50 | 2 | — | |
ZEGNZJNJHFUNKC
|
8.2 | IC50 | 2 | — | |
PNFAFGDVJIWRPA
|
7.9 | IC50 | 2 | — | |
UVEWXKOJMYQFGE
|
7.9 | IC50 | 2 | — | |
OKSIGHDJUXBCLG
|
7.9 | IC50 | 4 | — | |
BNSADWSGWCWEGZ
|
7.8 | IC50 | 2 | — | |
LDSDVQOOEYCWQS
|
7.8 | IC50 | 4 | — | |
FJLXFYHDLHZPQK
|
7.7 | IC50 | 4 | — | |
YSKANQRCYYKDSC
|
7.7 | IC50 | 4 | — | |
GSNXOPMMANYPOJ
|
7.7 | IC50 | 2 | — | |
FNFABWIIQJFQLF
|
7.7 | IC50 | 2 | — | |
BPCMQRINPLMHHT
|
7.6 | IC50 | 3 | — | |
NQWWXDNNFGCNQQ
|
7.5 | IC50 | 2 | — | |
UCTVTYJFSKGOLP
|
7.5 | IC50 | 2 | — | |
KJKVPMRFUZKTEA
|
7.5 | IC50 | 3 | — | |
CGYMRGTYHRRNMJ
|
7.5 | IC50 | 3 | — | |
JOWNADRSJZHOEJ
|
7.5 | IC50 | 2 | — | |
VQBICUVJQVNKBH
|
7.4 | IC50 | 4 | — | |
MLQJIASFGMOPPF
|
7.3 | IC50 | 2 | — | |
CFIJGRZCZVNJQK
|
7.2 | IC50 | 2 | — | |
MQVSMJMODJEBMM
|
7.2 | IC50 | 4 | — | |
AVFIHINZEZRGBL
|
7.2 | IC50 | 4 | — | |
OIYYXEBKWAWQQR
|
7.2 | IC50 | 2 | — | |
JMAUMLMBIAXZPR
|
7.2 | IC50 | 4 | — | |
LAGKZFNQXIBSDJ
|
7.2 | IC50 | 4 | — | |
NLYFSJWBMSCWSU
|
7.1 | IC50 | 4 | — | |
RLRGPZGIQMEBLC
|
7.1 | IC50 | 4 | — | |
BSWSHYUVWCPTHU
|
7.1 | IC50 | 4 | — | |
CYMWJZQYPTVZRX
|
7.1 | IC50 | 4 | — | |
IDVBVEOFBRZZEI
|
7.0 | IC50 | 5 | — | |
PSOBPHXKKHPWMU
|
7.0 | IC50 | 10 | — | |
VTUTUCVVSXMISL
|
7.0 | IC50 | 3 | — | |
ZMBZYRJHWCFIQA
|
7.0 | IC50 | 2 | — | |
ZNWWSWJQMFNZDV
|
7.0 | IC50 | 5 | — | |
QOMJHYUHYMCFHT
|
7.0 | IC50 | 4 | — | |
XSMABFRQESMONQ
|
7.0 | IC50 | 5 | — | |
VEDMWPYTXDSWTP
|
7.0 | IC50 | 4 | — | |
XWSGXVMUELGWLQ
|
7.0 | IC50 | 4 | — | |
RNTSNXOXDNEYJK
|
6.9 | IC50 | 4 | — | |
FQYVJQRHNLIPIK
|
6.9 | IC50 | 4 | — | |
GJJYDKIRDHZBBF
|
6.9 | IC50 | 2 | — | |
XAXOYJMMDIYHQF
|
6.9 | IC50 | 4 | — | |
MIHKHZZRKYZHJU
|
6.9 | IC50 | 4 | — | |
WQXQGYTXHBAVJS
|
6.9 | IC50 | 4 | — | |
ZBLHURFMYIWFIY
|
6.9 | IC50 | 4 | — | |
JRDMCDIQZVMPPB
|
6.9 | IC50 | 4 | — | |
AYSIHEFQSAIYGY
|
6.9 | IC50 | 4 | — | |
UZFOOEZHJLPYBL
|
6.9 | IC50 | 4 | — | |
BUTZNIHTVCLMKG
|
6.9 | IC50 | 4 | — |