Target Details
| UniProt AC | O75116 |
|---|---|
| Gene Symbol | ROCK2 |
| Protein Name | Rho-associated protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF25346 (PH_MRCK) PF00069 (Pkinase) PF08912 (Rho_Binding) |
Summary
- Multi-target molecules 1,696
- Clinical molecules 39
- Avg pChEMBL 7.47
KEGG Pathways (23)
- Adherens junction
- Axon guidance
- Cadherin signaling
- Chemokine signaling pathway
- Focal adhesion
- Human cytomegalovirus infection
- Leukocyte transendothelial migration
- Lipid and atherosclerosis
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Platelet activation
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Vascular smooth muscle contraction
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
- cGMP-PKG signaling pathway
Active Molecules (1,696)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LVAMWHFZQXITMS
|
7.9 | IC50 | 2 | — | |
QAJSUJQESOQFHQ
|
7.9 | IC50 | 2 | — | |
XGVDTEWKYAYOAZ
|
7.9 | IC50 | 2 | — | |
AWDORCFLUJZUQS
|
7.9 | IC50 | 7 | — | |
AXHOMFNSCRXCJW
|
7.9 | IC50 | 2 | — | |
CHSHJINQCNONGT
|
7.9 | IC50 | 2 | — | |
IQDPKFXHMNEJFH
|
7.9 | IC50 | 2 | — | |
LDNRNYZSQGXYFE
|
7.9 | IC50 | 2 | — | |
MPCRMOBUNIRDSJ
|
7.9 | IC50 | 2 | — | |
MQYQXIHEKOMMHJ
|
7.9 | IC50 | 2 | — | |
PJISZTIOUZPTEW
|
7.9 | IC50 | 2 | — | |
QOPVBHZKTCLPOW
|
7.9 | IC50 | 2 | — | |
SAGGCAPQVJYEGE
|
7.9 | IC50 | 3 | — | |
VUKPYAYVXNDTIK
|
7.9 | IC50 | 2 | — | |
ZPBGKGCPUCIWPT
|
7.9 | IC50 | 2 | — | |
ZRTWUBWXIGHVET
|
7.9 | IC50 | 2 | — | |
GWHBGZBCJKQNCZ
|
7.9 | IC50 | 4 | — | |
MXYAWDJBECRKLX
|
7.9 | IC50 | 6 | — | |
NVVLAIWWHAUHCF
|
7.9 | Ki | 4 | — | |
UHTJASDMENLSNM
|
7.9 | IC50 | 2 | — | |
ZMDKREPZDCSSGY
|
7.9 | IC50 | 2 | — | |
BLMKBLDBMAAGCC
|
7.9 | Ki | 3 | — | |
BSFNGHCTZDCQBF
|
7.9 | Ki | 93 | — | |
LUPCHAFIKZSOOK
|
7.9 | Ki | 15 | — | |
OORBXCUUHIIWJV
|
7.9 | IC50 | 2 | — | |
OUJZYQBEFNDJQN
|
7.9 | Ki | 71 | — | |
UFMAIBLTWQRHAK
|
7.9 | Ki | 10 | — | |
VIZWJTHWUUQVGO
|
7.9 | Ki | 9 | — | |
XSDJOIOVIMPMHD
|
7.9 | Ki | 44 | — | |
BVZFHBJXEPPCEX
|
7.9 | IC50 | 2 | — | |
GQMCGRYPKMDMGV
|
7.9 | IC50 | 2 | — | |
IFYDROJSRZHNOS
|
7.9 | IC50 | 7 | — | |
LBKUIYUPKQWTEX
|
7.9 | IC50 | 2 | — | |
NMVQKQZIFRBWNR
|
7.9 | IC50 | 2 | — | |
NZTPJNIILSLMRH
|
7.9 | IC50 | 7 | — | |
QXQGSOMQKZFIRY
|
7.9 | IC50 | 10 | — | |
UELSMLDRSQFVHG
|
7.9 | Ki | 4 | — | |
VIBAOTGKNYCAJL
|
7.9 | IC50 | 2 | — | |
WNDOFCPEDZYDPL
|
7.9 | IC50 | 10 | — | |
WPWSPITXILOZGO
|
7.9 | IC50 | 2 | — | |
WWFOLVBRNURGPW
|
7.9 | IC50 | 6 | — | |
YBJGEWMEAJHWTP
|
7.9 | IC50 | 2 | — | |
DXBVMSLBLNVYPE
|
7.9 | IC50 | 4 | — | |
PDSLHUWAGNRMJH
|
7.9 | IC50 | 2 | — | |
SCCMLQDEEDXQCZ
|
7.9 | Ki | 3 | — | |
YXAYEZQYTJGWNT
|
7.9 | IC50 | 2 | — | |
AQBIAGJFJKMCNG
|
7.8 | Ki | 4 | — | |
CAVXYZKAHQCDJF
|
7.8 | IC50 | 2 | — | |
GMLKJSOWCKBKLX
|
7.8 | IC50 | 5 | — | |
GVEIJKANJLOMJH
|
7.8 | IC50 | 2 | — |