Target Details
| UniProt AC | O60911 |
|---|---|
| Gene Symbol | CTSV |
| Protein Name | Cathepsin L2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 70
- Clinical molecules 0
- Avg pChEMBL 7.1
KEGG Pathways (2)
Active Molecules (70)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BWYBBMQLUKXECQ
|
10.2 | Ki | 5 | — | |
VBPPNJCVXGAZDD
|
8.7 | Ki | 5 | — | |
GXDULIFEODNFQZ
|
8.7 | IC50 | 4 | — | |
GXDULIFEODNFQZ
|
8.7 | IC50 | 4 | — | |
MFUOFOQCNPUGAP
|
8.5 | IC50 | 3 | — | |
MFUOFOQCNPUGAP
|
8.5 | IC50 | 3 | — | |
ACGFKLACOBPYKQ
|
8.2 | IC50 | 4 | — | |
ACGFKLACOBPYKQ
|
8.2 | IC50 | 4 | — | |
BPIZQAAUSWBFNS
|
8.2 | IC50 | 4 | — | |
BPIZQAAUSWBFNS
|
8.2 | IC50 | 4 | — | |
ZZDKLZGEJYCCFB
|
8.1 | IC50 | 4 | — | |
ZZDKLZGEJYCCFB
|
8.1 | IC50 | 4 | — | |
ABGBBQLBNIVODC
|
7.8 | IC50 | 4 | — | |
TXEWBLHLNYNUAG
|
7.7 | IC50 | 4 | — | |
TXEWBLHLNYNUAG
|
7.7 | IC50 | 4 | — | |
AVUGRCORGNXBOQ
|
7.6 | IC50 | 4 | — | |
AVUGRCORGNXBOQ
|
7.6 | IC50 | 4 | — | |
POELQXXPKHMGFF
|
7.5 | IC50 | 7 | — | |
CPDXLXNCBNKLMG
|
7.5 | IC50 | 4 | — | |
VKQOQWWJCCFELL
|
7.5 | IC50 | 4 | — | |
AEACXIXTPAQTGN
|
7.4 | IC50 | 4 | — | |
NVOCHHPUHMFGSJ
|
7.4 | IC50 | 4 | — | |
NVOCHHPUHMFGSJ
|
7.4 | IC50 | 4 | — | |
BKBPVMYBRCWYHF
|
7.2 | IC50 | 2 | — | |
BKBPVMYBRCWYHF
|
7.2 | IC50 | 2 | — | |
DFQDPBLCCLZOCK
|
7.2 | IC50 | 6 | — | |
LHHCSNFAOIFYRV
|
7.1 | IC50 | 8 | — | |
CDFSITIHQOZSIN
|
7.1 | IC50 | 7 | — | |
HYVXUIONWPXUDB
|
7.1 | IC50 | 4 | — | |
LBLSSIHBMJKAIZ
|
7.0 | Ki | 5 | — | |
NOMZQLLANMQZNR
|
7.0 | IC50 | 4 | — | |
NOMZQLLANMQZNR
|
7.0 | IC50 | 4 | — | |
IBVYZTXPOAZNHM
|
6.9 | IC50 | 3 | — | |
SIIJWJNEODXHNY
|
6.9 | IC50 | 7 | — | |
GCWIICJLIHIUNY
|
6.8 | IC50 | 7 | — | |
MNHLKDOPYXSVAC
|
6.8 | IC50 | 3 | — | |
MNHLKDOPYXSVAC
|
6.8 | IC50 | 3 | — | |
ZRKTXOUQLJMAQT
|
6.8 | IC50 | 3 | — | |
ZRKTXOUQLJMAQT
|
6.8 | IC50 | 3 | — | |
JPQIXMPQVCDFBY
|
6.8 | Ki | 5 | — | |
NFPHFQIUODNJRD
|
6.8 | IC50 | 5 | — | |
JKRUSRGXYHQECR
|
6.7 | IC50 | 3 | — | |
YKFSGPSMOHAYEG
|
6.7 | IC50 | 4 | — | |
HMVXEHSUUNUEBL
|
6.7 | IC50 | 4 | — | |
LTCAMZPTBRHGIT
|
6.7 | IC50 | 4 | — | |
MZRVIHRERYCHBL
|
6.7 | IC50 | 4 | — | |
XGRUEGXUKKXMFE
|
6.7 | IC50 | 3 | — | |
ZJUYWKXBSSDDNX
|
6.7 | IC50 | 3 | — | |
OGRMAGULSQOTTD
|
6.6 | Ki | 4 | — | |
SZYYBVWPURUFRR
|
6.6 | IC50 | 8 | — |