Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TUWDLUFFAHHNEF
|
7.6 | IC50 | 3 | — | |
UVCPBOQPPSLUPY
|
7.6 | IC50 | 3 | — | |
WQBRHFBWJUCVRR
|
7.6 | IC50 | 3 | — | |
XZYFNQNYLMTZIS
|
7.6 | IC50 | 3 | — | |
BXNOLMGJPGBWLA
|
7.6 | IC50 | 2 | — | |
CLMSQBWNXNAWOK
|
7.6 | IC50 | 2 | — | |
DCGPUMBJALMCLB
|
7.6 | IC50 | 3 | — | |
KPCAJGRRDIGSEF
|
7.6 | IC50 | 2 | — | |
NBBLMCRKPAWOPH
|
7.6 | IC50 | 3 | — | |
WKDIHLGAKPCUJV
|
7.6 | IC50 | 3 | — | |
XSISVIBLCIAEGR
|
7.6 | IC50 | 4 | — | |
BQDONWPMBNKZCG
|
7.6 | IC50 | 4 | — | |
FUOUPXXFTDVPGM
|
7.6 | IC50 | 3 | — | |
GPVRSQMGHNALCJ
|
7.6 | IC50 | 3 | — | |
IFLPDVNBLNGRJS
|
7.6 | IC50 | 3 | — | |
JBGZRMSDKXOUGQ
|
7.6 | IC50 | 2 | — | |
JKHAONFZTKWYFI
|
7.6 | IC50 | 2 | — | |
JKLFTZFZNNCDAE
|
7.6 | IC50 | 4 | — | |
KKQGFFSHWVTNMA
|
7.6 | IC50 | 3 | — | |
KQIUBFKRUFVQEI
|
7.6 | IC50 | 3 | — | |
LLRPIXCDTAUFLE
|
7.6 | IC50 | 4 | — | |
MLMDKPAWBXFXNA
|
7.6 | IC50 | 3 | — | |
PXLJQXYHONWMKB
|
7.6 | IC50 | 3 | — | |
RANSMASOMRJYFY
|
7.6 | IC50 | 2 | — | |
SFZBPQNERSUWOW
|
7.6 | IC50 | 3 | — | |
VJRCWRYAORRNAN
|
7.6 | IC50 | 2 | — | |
XQVVPGYIWAGRNI
|
7.6 | IC50 | 19 | — | |
FPGNUYNSOYSDAN
|
7.6 | IC50 | 2 | — | |
NZXJUZMTDGHZSR
|
7.6 | IC50 | 2 | — | |
CRXLFEZLSZPQMT
|
7.6 | IC50 | 2 | — | |
KGAKOIGDOIZZOQ
|
7.6 | IC50 | 2 | — | |
KLPMURBFDSDZSU
|
7.6 | IC50 | 3 | — | |
QSLHPKXGYOTUHN
|
7.6 | IC50 | 3 | — | |
UAEXWMVCHTWKPO
|
7.6 | IC50 | 2 | — | |
UJFLKMREHPPIRZ
|
7.6 | IC50 | 2 | — | |
BUFWGONUWXTMGP
|
7.6 | IC50 | 3 | — | |
BWMCWOZPWHUTGN
|
7.6 | IC50 | 3 | — | |
CMCDBYCMAWCMBJ
|
7.6 | IC50 | 2 | — | |
FDMPGPNYXCYCQJ
|
7.6 | IC50 | 3 | — | |
LSELSHXLKGXPPF
|
7.6 | Kd | 4 | — | |
NCNRHFGMJRPRSK
|
7.6 | IC50 | 14 | Yes | |
NWYXVTBJGUHMRR
|
7.6 | Kd | 3 | — | |
OFFYQYIVOWBZLD
|
7.6 | IC50 | 3 | — | |
PXTNXIAHIKBHPF
|
7.6 | IC50 | 3 | — | |
RKZATRLAMOOMLN
|
7.6 | IC50 | 2 | — | |
SKANTSCEPLCAJH
|
7.6 | IC50 | 2 | — | |
SKANTSCEPLCAJH
|
7.6 | IC50 | 2 | — | |
USNVRJYSAUJTNT
|
7.6 | IC50 | 4 | — | |
WSFUNVYDDZKPSU
|
7.6 | IC50 | 3 | — | |
LQNCVLFKDSYCTE
|
7.6 | IC50 | 2 | — |