Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FRDVUWTYVBTBSE
|
7.7 | IC50 | 3 | — | |
IGNHIECBXXHFPK
|
7.7 | IC50 | 2 | — | |
NHQWTZLQTWSZGU
|
7.7 | IC50 | 4 | — | |
OCOWZEOSBFUWRU
|
7.7 | IC50 | 2 | — | |
OEMGJZQIDXYGFV
|
7.7 | IC50 | 5 | — | |
PSWWDDSOCOGNCT
|
7.7 | IC50 | 2 | — | |
RIACYICSJAHABL
|
7.7 | Ki | 3 | — | |
RWRYTMPXTGYISG
|
7.7 | IC50 | 3 | — | |
SSELZXGQLGXCDT
|
7.7 | IC50 | 2 | — | |
SZLZPTHXIDWXLS
|
7.7 | Kd | 2 | — | |
TWYGARCNNFAUNW
|
7.7 | IC50 | 3 | — | |
YXHZTVCEXBXXJR
|
7.7 | IC50 | 3 | — | |
OIAZLVBSFCYPRC
|
7.7 | IC50 | 2 | — | |
ZGISYTAPMAPSIK
|
7.7 | IC50 | 3 | — | |
CBWCJYFVVHOTAZ
|
7.7 | Kd | 3 | — | |
FESHYOISGIZOBW
|
7.7 | IC50 | 2 | — | |
GPMKACUDCQFCCA
|
7.7 | IC50 | 2 | — | |
QCXJZVDATPNNCE
|
7.7 | IC50 | 3 | — | |
QUICABMRXTUSBQ
|
7.7 | IC50 | 2 | — | |
QXUMXOZTPSIGSM
|
7.7 | IC50 | 3 | — | |
SCLRZGNAIQFJNT
|
7.7 | IC50 | 3 | — | |
SXBROIQUJXJPJP
|
7.7 | IC50 | 3 | — | |
VLMANYNJKKOADM
|
7.7 | IC50 | 2 | — | |
WCNXRFKEDHKCLC
|
7.7 | IC50 | 3 | — | |
YJEIXSZAEKFWTM
|
7.7 | IC50 | 3 | — | |
BHEROPFARKLXOP
|
7.7 | IC50 | 4 | — | |
UYRUHHLEYUGTMC
|
7.7 | IC50 | 3 | — | |
AYMBFUSITNSKHY
|
7.6 | IC50 | 3 | — | |
CDERLIUJSXSXFH
|
7.6 | IC50 | 2 | — | |
GTLGKZJPNAWIBT
|
7.6 | IC50 | 3 | — | |
HQEUJXGKBKBFIW
|
7.6 | IC50 | 3 | — | |
JSKLBERKQHGHCP
|
7.6 | IC50 | 3 | — | |
KDVBPVJMVKBRPB
|
7.6 | IC50 | 2 | — | |
KJELUAWXBXCFLU
|
7.6 | IC50 | 2 | — | |
LMQMHIFIMOPETK
|
7.6 | IC50 | 3 | — | |
MRXGSXIGPZYETN
|
7.6 | IC50 | 3 | — | |
NCLGWTFZOQZNIS
|
7.6 | IC50 | 3 | — | |
RYGFKPUPLGKCHY
|
7.6 | IC50 | 3 | — | |
SSELZXGQLGXCDT
|
7.6 | IC50 | 3 | — | |
YGQMCJJLSQIPEF
|
7.6 | IC50 | 2 | — | |
YSAPPGXSSQEHTA
|
7.6 | IC50 | 3 | — | |
GAFAVXVVQUWUQX
|
7.6 | IC50 | 3 | — | |
VVPPHMRXPGDFBQ
|
7.6 | IC50 | 3 | — | |
CPWCZLPJMXCWDY
|
7.6 | IC50 | 3 | — | |
DVICYEUYFBDIJO
|
7.6 | IC50 | 3 | — | |
IYRDZCVNOKVDNI
|
7.6 | IC50 | 3 | — | |
KVTLTFKBEFZOGC
|
7.6 | IC50 | 3 | — | |
NRKGWEXMFVBBBE
|
7.6 | IC50 | 3 | — | |
OZSRLNZYSOUOCT
|
7.6 | IC50 | 3 | — | |
RLAHXCWDADVADO
|
7.6 | IC50 | 4 | — |