Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PXGREUPWZAUELV
|
7.8 | IC50 | 3 | — | |
QFTDPMPFNQAJTK
|
7.8 | Ki | 3 | — | |
QMWODUXCOTUXJT
|
7.8 | IC50 | 3 | — | |
SNIKOFNWYKITGY
|
7.8 | IC50 | 3 | — | |
STCCXFZWQGBXJD
|
7.8 | IC50 | 2 | — | |
SVEGTFMYOXJKMY
|
7.8 | IC50 | 3 | — | |
UAQDCZFGBBSHLT
|
7.8 | Kd | 4 | — | |
ZTGCZUISBHLGKD
|
7.8 | IC50 | 2 | — | |
AIEAYHRNULRMLO
|
7.8 | IC50 | 2 | — | |
FOEVWVKNXOCNTG
|
7.8 | IC50 | 3 | — | |
OOGDOIHBGKKMQF
|
7.8 | IC50 | 3 | — | |
VRVWHAZIBGEPEK
|
7.8 | Kd | 2 | — | |
ACNYFFICYHWMRO
|
7.7 | IC50 | 2 | — | |
AVWFNEVSOVPOLY
|
7.7 | IC50 | 3 | — | |
BUFWGONUWXTMGP
|
7.7 | IC50 | 3 | — | |
DVEBRKLPVWPNPS
|
7.7 | Kd | 2 | — | |
FKTRRXZUNCKQOU
|
7.7 | IC50 | 3 | — | |
JAXAHBJRANHVLF
|
7.7 | IC50 | 2 | — | |
LMBQVBQBODBFRL
|
7.7 | IC50 | 2 | — | |
MGLUYQBSWDKFIR
|
7.7 | IC50 | 3 | — | |
SCOGYYPZUPWMLU
|
7.7 | IC50 | 3 | — | |
WEHPZXXDBNJUIG
|
7.7 | IC50 | 3 | — | |
XMRBIQDRTZCVGG
|
7.7 | IC50 | 3 | — | |
XTJGRKJBJUZZJT
|
7.7 | IC50 | 2 | — | |
SWZWWWDWBVBZDV
|
7.7 | IC50 | 3 | — | |
VCBPMLSHIWJBBD
|
7.7 | IC50 | 2 | — | |
HNJGEQPWIDZIRC
|
7.7 | IC50 | 3 | — | |
MVALXNVRFKZEQJ
|
7.7 | IC50 | 2 | — | |
NMPGZGXWNHOBFF
|
7.7 | IC50 | 3 | — | |
RIDHDDTVNQHKEQ
|
7.7 | IC50 | 3 | — | |
RPBWYZZANXCAJX
|
7.7 | IC50 | 3 | — | |
UCTNVNGRNJPSOM
|
7.7 | IC50 | 3 | — | |
UXFXOEGGFKVCDW
|
7.7 | IC50 | 4 | — | |
WGJDGQSSFHDLIX
|
7.7 | IC50 | 3 | — | |
YMNUDRQQJNPPKD
|
7.7 | IC50 | 2 | — | |
AMRTUWDHDGIYSC
|
7.7 | IC50 | 3 | — | |
RGHQRULWHKEQHE
|
7.7 | IC50 | 3 | — | |
BRAMSTZRKUJRKS
|
7.7 | IC50 | 4 | — | |
GLMGIYSAZNFOHX
|
7.7 | IC50 | 3 | — | |
JVFXPRFAZLSBIF
|
7.7 | IC50 | 2 | — | |
KILRLNJOBPEYAV
|
7.7 | IC50 | 3 | — | |
LKEGXJXRNBALBV
|
7.7 | IC50 | 5 | — | |
LPZBOHUHUQVYMM
|
7.7 | IC50 | 2 | — | |
MNDAWZZJIIHLSL
|
7.7 | IC50 | 2 | — | |
NDEORODKVUYMFQ
|
7.7 | Kd | 9 | — | |
REHHQXJAWXFUSZ
|
7.7 | IC50 | 3 | — | |
YJEIXSZAEKFWTM
|
7.7 | IC50 | 3 | — | |
ZEBAQXYAFDJKJH
|
7.7 | IC50 | 2 | — | |
ZYJNOYAZLFPWBD
|
7.7 | IC50 | 4 | — | |
ZFJHDWKVFUWKQS
|
7.7 | IC50 | 3 | — |