Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GQVNARRVGGOXNP
|
7.8 | IC50 | 3 | — | |
GTYWOEFUZYKPQR
|
7.8 | IC50 | 3 | — | |
JBWFCYLPISSKIG
|
7.8 | IC50 | 3 | — | |
KQIUBFKRUFVQEI
|
7.8 | IC50 | 3 | — | |
NCLGWTFZOQZNIS
|
7.8 | IC50 | 3 | — | |
NEOVBISHUWMCQM
|
7.8 | IC50 | 3 | — | |
PKWSPAGTIXNWLL
|
7.8 | IC50 | 3 | — | |
QBWYZTMYCRAFMA
|
7.8 | Ki | 3 | — | |
QDMDJWBTMQQUPC
|
7.8 | IC50 | 3 | — | |
QMIQDDJVGIKUJA
|
7.8 | IC50 | 2 | — | |
QXTRPBVVUWEMOH
|
7.8 | IC50 | 2 | — | |
RFDBAEYXGSDEIK
|
7.8 | IC50 | 3 | — | |
YDFGIFLYGLMJSV
|
7.8 | IC50 | 4 | — | |
YQBHYHXPBGOPAY
|
7.8 | IC50 | 2 | — | |
YSAPPGXSSQEHTA
|
7.8 | IC50 | 3 | — | |
AWMLOQKKXSCDOQ
|
7.8 | IC50 | 2 | — | |
CBNDXTMVECMPGV
|
7.8 | IC50 | 4 | — | |
CHBGVONAUISDSX
|
7.8 | IC50 | 3 | — | |
CSMGGKQPASRAIQ
|
7.8 | IC50 | 3 | — | |
CYZNNGBIFDNKBV
|
7.8 | IC50 | 2 | — | |
DGXUFGAFFVEFEU
|
7.8 | IC50 | 3 | — | |
DVNSWDWISPDNHZ
|
7.8 | IC50 | 3 | — | |
FLEGAAQBQHISDY
|
7.8 | IC50 | 3 | — | |
HMRUYZVXBSSKBX
|
7.8 | IC50 | 3 | — | |
KDRSWORUPZEOGX
|
7.8 | IC50 | 3 | — | |
KHQQNXFBTALTQF
|
7.8 | IC50 | 6 | — | |
LDQWWSKUZGJSPQ
|
7.8 | IC50 | 2 | — | |
MGLUYQBSWDKFIR
|
7.8 | IC50 | 3 | — | |
OGOHNIGBBSGMEG
|
7.8 | IC50 | 2 | — | |
OSOMHZBGIZCTKM
|
7.8 | IC50 | 4 | — | |
PDCBJZVPIGAEBL
|
7.8 | IC50 | 4 | — | |
PVOCQBDIXSGBCZ
|
7.8 | IC50 | 2 | — | |
SCYBDERMEWGYSR
|
7.8 | IC50 | 2 | — | |
WZQLVEPIBAOOGF
|
7.8 | IC50 | 9 | — | |
XLAWIKASUIIZGC
|
7.8 | IC50 | 2 | — | |
GNMUEVRJHCWKTO
|
7.8 | IC50 | 3 | — | |
IBRUPFNOCSUECL
|
7.8 | IC50 | 3 | — | |
BYCJBYOKDKPJQP
|
7.8 | IC50 | 3 | — | |
DHQSSAHSRGVRJY
|
7.8 | IC50 | 3 | — | |
FFQNMMPQMYKTRZ
|
7.8 | Ki | 3 | — | |
GGRCIHACOIMRKY
|
7.8 | Ki | 2 | — | |
IAYAEBUJIVBSPF
|
7.8 | IC50 | 2 | — | |
IZWQPEYVFYWESQ
|
7.8 | IC50 | 3 | — | |
KKLVVGZXBWABFO
|
7.8 | IC50 | 3 | — | |
LEMUMFMXNFTRTL
|
7.8 | IC50 | 3 | — | |
NAPOLFVZKFHOBG
|
7.8 | IC50 | 4 | — | |
NLHZWVYLQRZHDF
|
7.8 | Ki | 3 | — | |
NSHYAULTAMQMBT
|
7.8 | IC50 | 2 | — | |
OMLHQPIYXLWGGG
|
7.8 | IC50 | 3 | — | |
PKHUSSXCMLLVRI
|
7.8 | IC50 | 3 | — |