Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYJCDALAOYQCIB
|
7.9 | IC50 | 2 | — | |
ZLVIFBCNFIAMBN
|
7.9 | IC50 | 3 | — | |
ZZJIAOWVSKZQGQ
|
7.9 | IC50 | 3 | — | |
DDSHVVXWYKDTTQ
|
7.9 | IC50 | 2 | — | |
SBOSVLRBKPEZMQ
|
7.9 | IC50 | 3 | — | |
AVWFNEVSOVPOLY
|
7.9 | IC50 | 3 | — | |
DDRRENHDNHGPEG
|
7.9 | IC50 | 3 | — | |
DVNSWDWISPDNHZ
|
7.9 | IC50 | 3 | — | |
HKDZBPLAJAVDDD
|
7.9 | IC50 | 2 | — | |
KJSPRHSFQGRYOT
|
7.9 | IC50 | 3 | — | |
LZQJKADDYCLNSB
|
7.9 | IC50 | 2 | — | |
NGGZYQVCSSIVJR
|
7.9 | IC50 | 2 | — | |
NMPGZGXWNHOBFF
|
7.9 | IC50 | 3 | — | |
NPLFXOGRUJPLAA
|
7.9 | IC50 | 3 | — | |
RCXOWIAUDIGVEW
|
7.9 | IC50 | 2 | — | |
RCXOWIAUDIGVEW
|
7.9 | IC50 | 2 | — | |
RJPKAAVNTLYQAC
|
7.9 | IC50 | 3 | — | |
UOBPZZRNSLHSFO
|
7.9 | IC50 | 2 | — | |
VFDAORCFAAAXRV
|
7.9 | IC50 | 3 | — | |
VLVRBRZAFGCGJV
|
7.9 | IC50 | 3 | — | |
VSKQFDSORJPDSV
|
7.9 | IC50 | 2 | — | |
WVDZBUCUXBEFHG
|
7.9 | IC50 | 3 | — | |
ZWXIRPBQXSHODB
|
7.9 | IC50 | 2 | — | |
KVKRYCAWRGWYNN
|
7.9 | IC50 | 3 | — | |
ZPZTZOURCDUBLM
|
7.9 | IC50 | 5 | — | |
FBYKSRDDFYPNNO
|
7.9 | IC50 | 3 | — | |
MDRXOFSNECSECW
|
7.9 | Kd | 4 | — | |
NECWWYRRULAEDN
|
7.9 | IC50 | 2 | — | |
BYVIHYLKGUPNHK
|
7.8 | IC50 | 3 | — | |
DMSRRTGRIHHJKS
|
7.8 | IC50 | 4 | — | |
FCGVFJQTWYBUCE
|
7.8 | IC50 | 2 | — | |
GVSWCHHMYQOERK
|
7.8 | IC50 | 2 | — | |
JMENTVKUBOUMCJ
|
7.8 | IC50 | 3 | — | |
JRPLDEULPIHXGO
|
7.8 | IC50 | 3 | — | |
OGJPTYDTRCDEJC
|
7.8 | IC50 | 3 | — | |
OGVXCCMPKKUNFP
|
7.8 | IC50 | 3 | — | |
PTLRUSZADXPAID
|
7.8 | IC50 | 2 | — | |
RGKUFEQXYKVMOO
|
7.8 | IC50 | 4 | — | |
RJDVRXGILIWOCC
|
7.8 | IC50 | 2 | — | |
UQMYMWRETIHSGQ
|
7.8 | IC50 | 3 | — | |
XMRBIQDRTZCVGG
|
7.8 | IC50 | 3 | — | |
YAJRUKJDKBVQBZ
|
7.8 | IC50 | 3 | — | |
JETVWIPZDARZAN
|
7.8 | IC50 | 3 | — | |
RSMYFSPOTCDHHJ
|
7.8 | IC50 | 5 | — | |
ZDMWQHIIHYYGIB
|
7.8 | IC50 | 3 | — | |
RGNILOZPZGAEOE
|
7.8 | IC50 | 2 | — | |
CUVAZMTZHFSHFL
|
7.8 | IC50 | 2 | — | |
CWBUVSFBCHVOPH
|
7.8 | Kd | 2 | — | |
FZOWBAIZBAZQAF
|
7.8 | IC50 | 2 | — | |
GLMGIYSAZNFOHX
|
7.8 | IC50 | 3 | — |