Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SJMFHBQDKBQDTQ
|
8.1 | IC50 | 2 | — | |
SJMFHBQDKBQDTQ
|
8.1 | IC50 | 2 | — | |
TUSWVDDMTVUGBQ
|
8.1 | IC50 | 2 | — | |
UACQAGADNJRGFK
|
8.1 | IC50 | 2 | — | |
UIWJGKYIPQKBHV
|
8.1 | IC50 | 4 | — | |
XBNRWYDSWFHTJI
|
8.1 | IC50 | 3 | — | |
XYXCJLYWFUGRHO
|
8.1 | Ki | 3 | — | |
YMNBDQGRLMZZPM
|
8.1 | IC50 | 2 | — | |
YYAYEFOQKNFTPU
|
8.1 | IC50 | 2 | — | |
QKJZSKDMERAPEK
|
8.0 | Kd | 2 | — | |
QSRRNUBIKNVQHO
|
8.0 | IC50 | 4 | — | |
SNBMTDIABWCKJS
|
8.0 | IC50 | 2 | — | |
WOHZTCPWKXURKU
|
8.0 | IC50 | 2 | — | |
BLPQMWXVHZTOMY
|
8.0 | IC50 | 2 | — | |
CNWQYJUFUYBRNG
|
8.0 | IC50 | 2 | — | |
PXHFZHKBGPQRAX
|
8.0 | IC50 | 2 | — | |
QUGZCQSQJAUOTO
|
8.0 | Ki | 3 | — | |
UIWJGKYIPQKBHV
|
8.0 | IC50 | 4 | — | |
YYKYSROKVREYAZ
|
8.0 | IC50 | 4 | — | |
ZJXAVKZXYZJJKO
|
8.0 | IC50 | 3 | — | |
ZZJIAOWVSKZQGQ
|
8.0 | IC50 | 3 | — | |
FXBLOXPPYWAJKD
|
8.0 | IC50 | 2 | — | |
RBZRCEPYYVFROZ
|
8.0 | Kd | 5 | — | |
ANEIGZBWQSTBKO
|
8.0 | IC50 | 2 | — | |
HMNJUXRTSGUSFM
|
8.0 | IC50 | 3 | — | |
JBPWXWQIGDWQHR
|
8.0 | IC50 | 15 | — | |
QHJUZMRVSGPOMP
|
8.0 | IC50 | 2 | — | |
RDWRDUFEWMSPGQ
|
8.0 | Kd | 4 | — | |
RIDHDDTVNQHKEQ
|
8.0 | IC50 | 3 | — | |
RKPWYUDCZHEUBU
|
8.0 | IC50 | 4 | — | |
VBNIZIAZOQSIGW
|
8.0 | IC50 | 2 | — | |
YORKSQKTPMJQBD
|
8.0 | IC50 | 3 | — | |
YPXANNJXRXDMDY
|
8.0 | Ki | 3 | — | |
URJBVMXNPKFWPB
|
8.0 | IC50 | 2 | — | |
WSHVXKCBHNIVJO
|
8.0 | IC50 | 4 | — | |
GHHBKDUDXQGYHF
|
7.9 | IC50 | 2 | — | |
MVALXNVRFKZEQJ
|
7.9 | IC50 | 2 | — | |
ASOYBTGQKMWPGU
|
7.9 | IC50 | 3 | — | |
CRYAUTCZOKUESS
|
7.9 | IC50 | 2 | — | |
DZUPEOBGVVEOJA
|
7.9 | Ki | 3 | — | |
IPYPJQJYDYFZCL
|
7.9 | IC50 | 3 | — | |
KJMPMBQYOMBJLE
|
7.9 | IC50 | 3 | — | |
KVPRUGZKNCVUEL
|
7.9 | IC50 | 2 | — | |
LAXUANUISYQZNT
|
7.9 | IC50 | 2 | — | |
NQGWNAPGXNVYHS
|
7.9 | IC50 | 3 | — | |
PBUQLYYLOVDBLR
|
7.9 | IC50 | 3 | — | |
RJVJSMKBCOIXKN
|
7.9 | IC50 | 3 | — | |
RZJAOODRKRAJBF
|
7.9 | IC50 | 2 | — | |
SADKUQHRGVTPSQ
|
7.9 | IC50 | 4 | — | |
WIHQCRGWXGPCAU
|
7.9 | IC50 | 2 | — |