Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GCDAPUPAGHUHLH
|
8.4 | IC50 | 4 | — | |
GCDAPUPAGHUHLH
|
8.4 | IC50 | 4 | — | |
PWEXGFMQMFFMNN
|
8.4 | IC50 | 4 | — | |
KTPZIQXMURKYQT
|
8.4 | IC50 | 2 | — | |
CJHOZKNBDTVZRM
|
8.3 | IC50 | 2 | — | |
DCXAWDGRFZGDMY
|
8.3 | IC50 | 2 | — | |
ICUFVYYLUGJQPU
|
8.3 | IC50 | 2 | — | |
UUCXBSUBBNYHGE
|
8.3 | IC50 | 2 | — | |
WBGMNYXQTDAOTN
|
8.3 | IC50 | 2 | — | |
VEPYYWIOIMZOLX
|
8.3 | IC50 | 4 | — | |
IQSNRFQUNLCFPX
|
8.3 | IC50 | 2 | — | |
KBHPDJCNCCZDFQ
|
8.3 | IC50 | 2 | — | |
RJJDAOYTHRXSGL
|
8.3 | IC50 | 4 | — | |
UIINOGWJPAPJTM
|
8.3 | IC50 | 2 | — | |
VYNYPLNNLNISCK
|
8.3 | IC50 | 4 | — | |
XBGAIUVLEXZQMO
|
8.2 | IC50 | 4 | — | |
XQSIYYHBLOKYON
|
8.2 | IC50 | 2 | — | |
FAWSUKOIROHXAP
|
8.2 | IC50 | 5 | — | |
SOKDPRRREPVZBP
|
8.2 | IC50 | 2 | — | |
CIDSGDKXNGKZIH
|
8.2 | IC50 | 2 | — | |
WSYLTXUNMXZHLY
|
8.2 | IC50 | 2 | — | |
XBGAIUVLEXZQMO
|
8.2 | IC50 | 4 | — | |
QWAOMERKQXGSJH
|
8.2 | IC50 | 2 | — | |
MFKPAAFGGBINQO
|
8.2 | IC50 | 4 | — | |
TUDWFCNTNUMOKQ
|
8.2 | IC50 | 2 | — | |
WQOHYQKCKHFIMI
|
8.2 | IC50 | 2 | — | |
HSAHLMIFPRYVEH
|
8.2 | IC50 | 4 | — | |
SJLGONPWSYKHIB
|
8.2 | IC50 | 2 | — | |
UDJIOTIVUUWIDN
|
8.2 | IC50 | 2 | — | |
WUJOUMVRCGTKNK
|
8.2 | IC50 | 2 | — | |
XXMVJVPJGYCSFZ
|
8.2 | IC50 | 2 | — | |
CWTFXHWWWKKEQI
|
8.1 | Kd | 2 | — | |
GSWRJJUJRPXSPR
|
8.1 | IC50 | 3 | — | |
XXARZBLNZNGJPR
|
8.1 | IC50 | 2 | — | |
PQOGZKGXGLHDGS
|
8.1 | Kd | 4 | — | |
FBYKSRDDFYPNNO
|
8.1 | IC50 | 3 | — | |
DHJBCEVAMQVGRX
|
8.1 | IC50 | 2 | — | |
FSVRQKKTQOWUTB
|
8.1 | IC50 | 2 | — | |
IEVUMROHFZOVMK
|
8.1 | IC50 | 3 | — | |
IJZDKKQZNSYLGO
|
8.1 | IC50 | 2 | — | |
KMDXJEQFNWVGIH
|
8.1 | Ki | 3 | — | |
OMVCEOIEFNQPMM
|
8.1 | IC50 | 2 | — | |
WEGRDNGNIKWFOP
|
8.1 | IC50 | 2 | — | |
AEANZCXROGPSBY
|
8.1 | Ki | 6 | — | |
FQVGCUZGXCCGOC
|
8.1 | IC50 | 2 | — | |
RCDQFASKGQECOZ
|
8.1 | Ki | 2 | — | |
WSOSPNZDGBUARC
|
8.1 | IC50 | 2 | — | |
BCOBWZAGQAFMQP
|
8.1 | IC50 | 2 | — | |
CAFIQDSDKILBAO
|
8.1 | IC50 | 2 | — | |
JLUUVUUYIXBDCG
|
8.1 | IC50 | 2 | — |