Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OPRLJTKXGDBVAC
|
8.7 | IC50 | 2 | — | |
OTLUGLDCVHKZEE
|
8.7 | IC50 | 2 | — | |
QCVBUWRWHOLCOJ
|
8.7 | IC50 | 2 | — | |
RKCDVGZWRITJMS
|
8.7 | IC50 | 2 | — | |
RPOVNYLBJCXTOQ
|
8.7 | IC50 | 2 | — | |
RZNVPBJTIYRMSE
|
8.7 | IC50 | 2 | — | |
UOGTVNXJONPDSD
|
8.7 | IC50 | 2 | — | |
QDOKVLKQKZPGPG
|
8.6 | IC50 | 2 | — | |
UETQFSCWDMJWMM
|
8.6 | IC50 | 4 | — | |
JNYHQYRTYFSMSQ
|
8.6 | IC50 | 3 | — | |
LOOFPBVYOVHBCL
|
8.5 | IC50 | 3 | — | |
AIFXAXRMMBWMAG
|
8.5 | Kd | 4 | — | |
AMHWRJBEKUEFFO
|
8.5 | Kd | 2 | — | |
BFYPTOVDLGDJDC
|
8.5 | IC50 | 2 | — | |
BMBTWLMYKIAXLA
|
8.5 | IC50 | 2 | — | |
CUQCNMCZQPPDII
|
8.5 | IC50 | 2 | — | |
ICGXDGBYQZIXIF
|
8.5 | IC50 | 2 | — | |
MJCKFIWZHNIKPQ
|
8.5 | Kd | 2 | — | |
NYYNLDHMWIENMY
|
8.5 | IC50 | 2 | — | |
OJPOVVTUDJNUND
|
8.5 | IC50 | 2 | — | |
OYPQYGXUQANMSS
|
8.5 | IC50 | 2 | — | |
PWPYJSVOLAVRNB
|
8.5 | IC50 | 2 | — | |
QQUFYDKFQLICRA
|
8.5 | IC50 | 2 | — | |
RDONXGFGWSSFMY
|
8.5 | IC50 | 6 | — | |
VUUYIKCADVQZHC
|
8.5 | IC50 | 2 | — | |
RZUVKPXJAZFJJR
|
8.5 | IC50 | 2 | — | |
DPQKUYBPPCXREN
|
8.5 | Kd | 2 | — | |
OEDSFMUSNZDJFD
|
8.5 | Ki | 4 | — | |
WEQSOZXIXPNDJW
|
8.5 | IC50 | 2 | — | |
WOSYEWDDCNUUHT
|
8.5 | IC50 | 4 | — | |
ONTCKBVHGQBHTF
|
8.5 | IC50 | 3 | — | |
SFYLADBQGNFSOV
|
8.5 | IC50 | 2 | — | |
VQOLNDHLOBZXNA
|
8.5 | IC50 | 2 | — | |
FNHHVPPSBFQMEL
|
8.4 | IC50 | 4 | — | |
LMYMWXJBPLXESU
|
8.4 | Kd | 2 | — | |
YTJRGAPMTDBXIK
|
8.4 | Kd | 2 | — | |
PWFGHENEZLVBOP
|
8.4 | Kd | 2 | — | |
BJGCRXAPTHEXLQ
|
8.4 | IC50 | 2 | — | |
BVNSMRUDPSJEIU
|
8.4 | IC50 | 2 | — | |
FCQIYPQMTYFWQM
|
8.4 | IC50 | 2 | — | |
FYSWLIFIYIVHPI
|
8.4 | Kd | 4 | — | |
HWYPQYNAVWQEKO
|
8.4 | IC50 | 2 | — | |
NFMDDLDYDOZPGW
|
8.4 | IC50 | 2 | — | |
OJSKWCXPUVTNCF
|
8.4 | IC50 | 4 | — | |
UMQADUCCACBHKD
|
8.4 | IC50 | 2 | — | |
VBRWZRVQWASOOS
|
8.4 | IC50 | 2 | — | |
VLSNXLPXZLYNBB
|
8.4 | IC50 | 2 | — | |
WIXBOVBNLLVASA
|
8.4 | IC50 | 2 | — | |
XYVCWEWEPXYPNF
|
8.4 | IC50 | 2 | — | |
ZHQPTIFREKVURJ
|
8.4 | IC50 | 2 | — |