Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DLOWILGTRNUHPQ
|
7.0 | Kd | 2 | — | |
HKECFOZBEGKIAX
|
7.0 | IC50 | 3 | — | |
KRBXHYJZXGUPRJ
|
7.0 | IC50 | 3 | — | |
MWVVALQFXSOQLF
|
7.0 | IC50 | 3 | — | |
OVLDCYAZEIXCEQ
|
7.0 | IC50 | 4 | — | |
OYLZIDSUJMGMBF
|
7.0 | IC50 | 3 | — | |
QUMCIHKVKQYNPA
|
7.0 | IC50 | 2 | — | |
RTFLOGJKYBGANO
|
7.0 | IC50 | 4 | — | |
UFJLBLXSGFZNIM
|
7.0 | IC50 | 2 | — | |
XPDXANVGYAEATN
|
7.0 | IC50 | 3 | — | |
YGQSAYAQCWLSAL
|
7.0 | IC50 | 3 | — | |
YINBDXKXEYUKBO
|
7.0 | IC50 | 3 | — | |
INSOERIUGCDMID
|
7.0 | IC50 | 2 | — | |
KDPQFXRDUUVUMM
|
6.9 | IC50 | 2 | — | |
KXEMGSZLUNPCML
|
6.9 | IC50 | 2 | — | |
QIEVBHRUPLMWFP
|
6.9 | IC50 | 2 | — | |
UYBRROMMFMPJAN
|
6.9 | IC50 | 8 | — | |
YCNMRNSZEJLPCH
|
6.9 | IC50 | 2 | — | |
ZYPRPLRGMSHRRW
|
6.9 | IC50 | 2 | — | |
IHOWNNYVAUSWOU
|
6.9 | IC50 | 7 | — | |
LMLJGVCFCYGAST
|
6.9 | IC50 | 3 | — | |
PTAMRJLIOCHJMQ
|
6.9 | Kd | 6 | — | |
RXAFLNFTNQFCIB
|
6.9 | IC50 | 2 | — | |
AMGMXABLUGQVQD
|
6.9 | IC50 | 3 | — | |
DUZXHNLPDHPTHC
|
6.9 | IC50 | 3 | — | |
GXKIVKDALCGWBS
|
6.9 | IC50 | 3 | — | |
HBIBLLVDGBUKCQ
|
6.9 | IC50 | 4 | — | |
IBJLUHJBIGMOMD
|
6.9 | IC50 | 4 | — | |
IPJMGURQBOGYIE
|
6.9 | IC50 | 4 | — | |
IPZXGSLENCVPEZ
|
6.9 | IC50 | 2 | — | |
IQIUDSWFPYGIST
|
6.9 | IC50 | 3 | — | |
IVGGZYPSQXBUGB
|
6.9 | IC50 | 2 | — | |
JBDVGVNIQOSQQT
|
6.9 | IC50 | 2 | — | |
KPXMSUZHJCHOTN
|
6.9 | Kd | 3 | — | |
LKHKHWRBQLPSBP
|
6.9 | IC50 | 3 | — | |
LRWGLQDVNJOJKQ
|
6.9 | IC50 | 3 | — | |
MTBDHPJCWYLCBM
|
6.9 | IC50 | 7 | — | |
MTKZUOYFXZHUDU
|
6.9 | IC50 | 3 | — | |
NVUCJVXTEMYIJR
|
6.9 | IC50 | 3 | — | |
RQCMHFWZGCIXKC
|
6.9 | IC50 | 2 | — | |
SXNJFOWDRLKDSF
|
6.9 | Kd | 8 | — | |
WHSDNSXIFWGGOD
|
6.9 | IC50 | 4 | — | |
WSQOJBUQSYKMGG
|
6.9 | IC50 | 2 | — | |
XFGHSUSRHXWNEX
|
6.9 | IC50 | 3 | — | |
XSOFZNARGSJIQN
|
6.9 | IC50 | 4 | — | |
ZAIFEOJGYZIMNX
|
6.9 | IC50 | 3 | — | |
FIMCUEFPUNBSJO
|
6.9 | IC50 | 2 | — | |
XXZLLCKEAYMUHY
|
6.9 | IC50 | 2 | — | |
AUXWZPVOQCZHSP
|
6.9 | IC50 | 2 | — | |
ISCJKSNXTHTNBW
|
6.9 | IC50 | 4 | — |