Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XYDZHZCXCJNSIB
|
7.0 | IC50 | 3 | — | |
YLEHNGYWUWDXNV
|
7.0 | IC50 | 3 | — | |
ZPMULUKHFNMJPF
|
7.0 | IC50 | 2 | — | |
FLLDFQACNKMSRM
|
7.0 | IC50 | 3 | — | |
JFPHLFWFVVJKQO
|
7.0 | IC50 | 4 | — | |
JSJHNZMAOMLIME
|
7.0 | IC50 | 3 | — | |
MZKIOOQWOZDDMX
|
7.0 | IC50 | 3 | — | |
NTQVJGUGYLGXNI
|
7.0 | IC50 | 3 | — | |
QECMENZMDBOLDR
|
7.0 | IC50 | 2 | — | |
QXYGIHZVXILREV
|
7.0 | IC50 | 3 | — | |
CFTIJALKSHXVNU
|
7.0 | IC50 | 3 | — | |
ONIDJCXYPGJIMN
|
7.0 | IC50 | 2 | — | |
PJFBYCXYSAXHLS
|
7.0 | IC50 | 2 | — | |
UNVPHVSVVHLLKD
|
7.0 | IC50 | 2 | — | |
ZPMULUKHFNMJPF
|
7.0 | IC50 | 2 | — | |
CFXFHVGCTLQYSO
|
7.0 | IC50 | 2 | — | |
IVXYIGADMWHQDD
|
7.0 | IC50 | 4 | — | |
KDQRDBUPLHFYBU
|
7.0 | IC50 | 2 | — | |
KUCAMLWGYMEYGQ
|
7.0 | IC50 | 3 | — | |
LBXYVUXGPFEVSI
|
7.0 | IC50 | 3 | — | |
NYYPYDLZLGCKOU
|
7.0 | IC50 | 4 | — | |
PASBWKAEFYVJHG
|
7.0 | IC50 | 3 | — | |
GEGMKHTYQVNYFV
|
7.0 | IC50 | 2 | — | |
JGGBFOUTSJEGRT
|
7.0 | Ki | 4 | — | |
KXSJLOFFUFDGTE
|
7.0 | IC50 | 6 | — | |
UXOOYKGHOJVFQB
|
7.0 | IC50 | 3 | — | |
VEUMTIQGKUVYJM
|
7.0 | IC50 | 2 | — | |
HDFQNQPMGAHQTL
|
7.0 | IC50 | 5 | — | |
ITQINGMSTPZGFO
|
7.0 | IC50 | 3 | — | |
OGSOMZCUMMDDJU
|
7.0 | IC50 | 4 | — | |
PMIMBFPXSMELLC
|
7.0 | IC50 | 3 | — | |
SDLMPYCGZKLARA
|
7.0 | IC50 | 4 | — | |
STEDHESXTGJFOX
|
7.0 | IC50 | 3 | — | |
SUNGCKMWYWAHPK
|
7.0 | IC50 | 3 | — | |
VVRZMYLMDPVHTL
|
7.0 | Ki | 3 | — | |
WUFYDWKEOKQEEP
|
7.0 | IC50 | 3 | — | |
HTYUJAPSAJUBKN
|
7.0 | IC50 | 2 | — | |
KLKMODXQLGKDKQ
|
7.0 | Ki | 3 | — | |
OSSMVMKSVHUBNI
|
7.0 | IC50 | 2 | — | |
PVDBPOSKQRWTRG
|
7.0 | IC50 | 3 | — | |
RJQMEGOXPKMDFQ
|
7.0 | IC50 | 2 | — | |
SBDOCCVDBJLSLR
|
7.0 | IC50 | 3 | — | |
VBDIOKSSYUZONA
|
7.0 | IC50 | 3 | — | |
VUVUVNZRUGEAHB
|
7.0 | IC50 | 5 | — | |
DYQPKOGFUIEBMS
|
7.0 | IC50 | 3 | — | |
IRCDNPBWELYZBD
|
7.0 | IC50 | 3 | — | |
JCGSQIXZALUTFO
|
7.0 | IC50 | 2 | — | |
SVWVGWHDUPYUFQ
|
7.0 | IC50 | 4 | — | |
BKDMSQCDGPSQFW
|
7.0 | IC50 | 3 | — | |
CWZBKMRDRUFOGI
|
7.0 | IC50 | 3 | — |