Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CPTTUKGIGKOQKE
|
7.1 | IC50 | 2 | — | |
FUXOAMWDPVPAFQ
|
7.1 | IC50 | 3 | — | |
IITSESCLMNYTBQ
|
7.1 | IC50 | 3 | — | |
IWELMDBRVJWCNU
|
7.1 | IC50 | 2 | — | |
LEXSRVMWXAFLMV
|
7.1 | IC50 | 4 | — | |
LHEGCVROQQOOOL
|
7.1 | IC50 | 3 | — | |
MXCCPOZZBZEVAU
|
7.1 | IC50 | 2 | — | |
QZZCUOVXHPAQRQ
|
7.1 | IC50 | 5 | — | |
SJSCJYHUBPKPNG
|
7.1 | IC50 | 3 | — | |
UBBQMWGFAITOCR
|
7.1 | IC50 | 2 | — | |
WCMQEPUDHFATFM
|
7.1 | Kd | 3 | — | |
AAFNIAPCKWGXDG
|
7.1 | IC50 | 3 | — | |
BFZZIGPNZLXGRV
|
7.1 | IC50 | 3 | — | |
DBBQRLYYNNWGPM
|
7.1 | Kd | 3 | — | |
FAMCYVZRWHZORW
|
7.1 | IC50 | 3 | — | |
MYTABVRHXGACGI
|
7.1 | IC50 | 4 | — | |
OFLADKRRSZHEFK
|
7.1 | IC50 | 2 | — | |
OOSHYWXSNYXCER
|
7.1 | IC50 | 2 | — | |
TYOPZGWEWQOLHM
|
7.1 | IC50 | 2 | — | |
DYQPKOGFUIEBMS
|
7.1 | IC50 | 3 | — | |
IWBBXOOPRPDUIL
|
7.1 | IC50 | 3 | — | |
LTGAYVZNSVTKFS
|
7.1 | IC50 | 3 | — | |
MSZSAGAHXQKHRZ
|
7.1 | IC50 | 3 | — | |
SDIHFORMFMHWNK
|
7.1 | IC50 | 6 | — | |
BWECVGNIEMDNMY
|
7.1 | IC50 | 2 | — | |
FLLDFQACNKMSRM
|
7.1 | IC50 | 3 | — | |
KGPRTZSROXHRIX
|
7.1 | IC50 | 2 | — | |
NVUCJVXTEMYIJR
|
7.1 | IC50 | 3 | — | |
STSKCRDOTKSTPF
|
7.1 | IC50 | 3 | — | |
UWHQJIJZHLHELR
|
7.1 | IC50 | 4 | — | |
VAXZYGLGDOWBGT
|
7.1 | IC50 | 3 | — | |
ZBZCQXDDHPHITA
|
7.1 | IC50 | 4 | — | |
ZQTWZFDWESQAJC
|
7.1 | IC50 | 4 | — | |
BNWMHKNZCUUJMF
|
7.1 | IC50 | 3 | — | |
DVMCRBPTCKGCAX
|
7.1 | IC50 | 2 | — | |
FSMTUHGXWGJNKK
|
7.1 | IC50 | 4 | — | |
FTHLNVOKHACXIU
|
7.1 | IC50 | 3 | — | |
FUOUPXXFTDVPGM
|
7.1 | IC50 | 3 | — | |
MHDJYXZJVBCMGS
|
7.1 | IC50 | 3 | — | |
MZPJSFUFCBJTIP
|
7.1 | IC50 | 2 | — | |
PUVZCXWHNDJBCX
|
7.1 | IC50 | 2 | — | |
SRFOIWNXIILSNJ
|
7.1 | IC50 | 4 | — | |
AJFFVWPPDGTGNY
|
7.0 | IC50 | 2 | — | |
FFHFKSXIZXKTRE
|
7.0 | IC50 | 3 | — | |
KDPQFXRDUUVUMM
|
7.0 | IC50 | 2 | — | |
OZPNRBXVIUPSDJ
|
7.0 | IC50 | 4 | — | |
PIWFRDGCNFFYEO
|
7.0 | IC50 | 3 | — | |
QKXLHLCDBNXSBT
|
7.0 | IC50 | 2 | — | |
QNRNHBQTJGHZSO
|
7.0 | IC50 | 3 | — | |
WVDZBUCUXBEFHG
|
7.0 | IC50 | 3 | — |