Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WCNXRFKEDHKCLC
|
7.2 | IC50 | 3 | — | |
YXEKBZDFBBBFJB
|
7.2 | IC50 | 2 | — | |
ZNGYYGUCWRDEAS
|
7.2 | IC50 | 3 | — | |
ZOVYOHAZPIKVOR
|
7.2 | IC50 | 4 | — | |
BNWMHKNZCUUJMF
|
7.2 | IC50 | 3 | — | |
IEEQBCSZMPIUGM
|
7.2 | IC50 | 3 | — | |
LCXHXIMNUYTCEI
|
7.2 | IC50 | 3 | — | |
MJNSUGCWCAGANT
|
7.2 | IC50 | 3 | — | |
PYJQEIWIODYCRH
|
7.2 | IC50 | 3 | — | |
WVPDDEACKJQZHD
|
7.2 | IC50 | 2 | — | |
XASDFFVVUGREBP
|
7.2 | IC50 | 3 | — | |
YXHZTVCEXBXXJR
|
7.2 | IC50 | 3 | — | |
ZQFOFTHJENGQKG
|
7.2 | IC50 | 3 | — | |
ASFZUTSSNARCOL
|
7.2 | IC50 | 3 | — | |
DDHSJBNVVYBOFE
|
7.2 | Kd | 2 | — | |
ICPNDBHZFPANIZ
|
7.2 | IC50 | 2 | — | |
IWMCPJZTADUIFX
|
7.2 | Kd | 3 | — | |
LYAOPUXRPJKSKW
|
7.2 | Kd | 3 | — | |
QZHPNAKQERGIOM
|
7.2 | IC50 | 2 | — | |
SAFUIPXIPYTSEU
|
7.2 | IC50 | 2 | — | |
SUIIIOQGACLJMI
|
7.2 | IC50 | 3 | — | |
AAAQFGUYHFJNHI
|
7.2 | IC50 | 252 | — | |
BHZGECKOYMLRSO
|
7.2 | IC50 | 3 | — | |
FEBAVJBCNBJJOC
|
7.2 | IC50 | 2 | — | |
FPKFEJQELSGORT
|
7.2 | IC50 | 2 | — | |
OSBPICGFSLCYPI
|
7.2 | IC50 | 2 | — | |
XDAXVUPUYYWFHA
|
7.2 | IC50 | 3 | — | |
ZBKQIKDKLUJFMK
|
7.2 | Ki | 3 | — | |
BHHISRQWOKUVFO
|
7.1 | IC50 | 3 | — | |
FTYXFBKWRBABJZ
|
7.1 | IC50 | 3 | — | |
GWHBOLQUVHIAPZ
|
7.1 | IC50 | 4 | — | |
NQROQCRXQDNZSD
|
7.1 | Kd | 3 | — | |
SJACAKNFJFXOJF
|
7.1 | IC50 | 3 | — | |
SSCBXXKTZLTDDN
|
7.1 | IC50 | 3 | — | |
GGZYNJKDGRBRKG
|
7.1 | IC50 | 2 | — | |
ICQWKYPGTXWGCR
|
7.1 | IC50 | 2 | — | |
JXLHJBYUGDELIZ
|
7.1 | IC50 | 2 | — | |
SWQSOOOMILGDNL
|
7.1 | IC50 | 2 | — | |
AWVPNUWHMBPXOU
|
7.1 | Kd | 8 | — | |
DQDVRWIYUXKYQR
|
7.1 | IC50 | 2 | — | |
GFDDTDKCZCGJLM
|
7.1 | Kd | 5 | — | |
URJQRGYKGNGARR
|
7.1 | IC50 | 2 | — | |
YHMNROQTPUKNLA
|
7.1 | IC50 | 8 | — | |
FQEWVABJRCOJBI
|
7.1 | IC50 | 3 | — | |
HXVTYKVZGFHITR
|
7.1 | IC50 | 3 | — | |
IMUJKGKBDBVTGZ
|
7.1 | IC50 | 3 | — | |
MPDWALFCXGTZJW
|
7.1 | IC50 | 3 | — | |
VUWJZAUOMZSUEU
|
7.1 | IC50 | 3 | — | |
WDADYPXHXOFAQY
|
7.1 | Kd | 2 | — | |
WQRKDXUDKMFKPL
|
7.1 | IC50 | 4 | — |