Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UZPOOTYPBOTHKT
|
7.2 | IC50 | 3 | — | |
XRYCKSUJUPLGRF
|
7.2 | IC50 | 2 | — | |
YJLPEIDBEOKJJP
|
7.2 | IC50 | 2 | — | |
BRBCSVDUUHHTIS
|
7.2 | IC50 | 4 | — | |
BVDVIORIEDCJPV
|
7.2 | IC50 | 3 | — | |
CFUYRGUSQPAALN
|
7.2 | IC50 | 3 | — | |
FNDFWBANYDEWBA
|
7.2 | Kd | 3 | — | |
XSORNHYQCJBFAK
|
7.2 | IC50 | 2 | — | |
BEEOECFSSLHUJR
|
7.2 | IC50 | 2 | — | |
CBIPLHJRIODVHF
|
7.2 | IC50 | 2 | — | |
DDIGBXFXYQBMSG
|
7.2 | IC50 | 3 | — | |
FLASGTNYMYVYKJ
|
7.2 | IC50 | 3 | — | |
GKJNYZBASPYBEP
|
7.2 | IC50 | 3 | — | |
HTPNGOWITIWAHM
|
7.2 | IC50 | 3 | — | |
HXENBKGGEPBXOQ
|
7.2 | IC50 | 3 | — | |
ZNKHCSORNQHLOY
|
7.2 | IC50 | 2 | — | |
HIZNONHBBUUYFX
|
7.2 | IC50 | 4 | — | |
KQUKQLUXCYAWHW
|
7.2 | IC50 | 2 | — | |
LBAXGISUFHVKPW
|
7.2 | IC50 | 2 | — | |
MJTVRIBROYBHIV
|
7.2 | IC50 | 3 | — | |
PLMVDZBEQUQDAZ
|
7.2 | IC50 | 2 | — | |
ULDFEUPLPPWJDA
|
7.2 | IC50 | 3 | — | |
AREGGTVPTLNTCU
|
7.2 | IC50 | 3 | — | |
CAKYNETUOQZPMX
|
7.2 | IC50 | 2 | — | |
HVCZNOOIHIEREB
|
7.2 | IC50 | 2 | — | |
LFNLJQQQSRYUHQ
|
7.2 | IC50 | 3 | — | |
RSTUWYLUVVSQFJ
|
7.2 | IC50 | 2 | — | |
RUHXXMHOKIHJKY
|
7.2 | IC50 | 2 | — | |
UZPOOTYPBOTHKT
|
7.2 | IC50 | 3 | — | |
XQSKFZQVORBNFZ
|
7.2 | IC50 | 2 | — | |
ZBKQSWPCHUEZBL
|
7.2 | IC50 | 3 | — | |
ARWMKZDWGIOCEU
|
7.2 | Kd | 4 | — | |
BHJOJVLBZYUYGS
|
7.2 | IC50 | 6 | — | |
GACUWBJOGWUMHF
|
7.2 | Kd | 2 | — | |
GQXFGAMRIGUNFT
|
7.2 | IC50 | 4 | — | |
KNBYFXZNSOENGW
|
7.2 | IC50 | 5 | — | |
MCVXORPOSRGRKJ
|
7.2 | IC50 | 2 | — | |
ODYIWGILJYUPOR
|
7.2 | IC50 | 3 | — | |
SGTKTGFQXONNJX
|
7.2 | IC50 | 2 | — | |
VWXSUJYWCXZAIC
|
7.2 | IC50 | 2 | — | |
XBQGLWPUGBREQS
|
7.2 | IC50 | 4 | — | |
YDIQBHXHQQZJQQ
|
7.2 | IC50 | 3 | — | |
OENGVXVRDHPNME
|
7.2 | IC50 | 3 | — | |
OTZHGAAUXLOJFP
|
7.2 | IC50 | 3 | — | |
QIJUHAIEZZEKSX
|
7.2 | IC50 | 3 | — | |
SKTNIECRSURWAZ
|
7.2 | IC50 | 3 | — | |
XNRZMTWJFLFRMR
|
7.2 | IC50 | 3 | — | |
HFXQHVKVUNQRBN
|
7.2 | IC50 | 7 | — | |
PXGREUPWZAUELV
|
7.2 | IC50 | 3 | — | |
PXGREUPWZAUELV
|
7.2 | IC50 | 3 | — |