Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZKANYDYIVJBAM
|
7.3 | IC50 | 2 | — | |
XOCKWBJNBUYYAL
|
7.3 | IC50 | 5 | — | |
ZLSFDTLLWMDEFA
|
7.3 | IC50 | 2 | — | |
ZUTVFNRARULPEX
|
7.3 | IC50 | 2 | — | |
KIGOYJHUPSVEGZ
|
7.3 | IC50 | 2 | — | |
ORTRBMKXQWFMTN
|
7.3 | IC50 | 3 | — | |
UBXNLHDUJFHNDS
|
7.3 | IC50 | 3 | — | |
WLWYLWZRQXMOQI
|
7.3 | IC50 | 2 | — | |
BIUDFTNJMGSWCJ
|
7.3 | IC50 | 2 | — | |
DNVXATUJJDPFDM
|
7.3 | IC50 | 17 | — | |
FRBRZGLUFOZRGD
|
7.3 | IC50 | 5 | — | |
FRBRZGLUFOZRGD
|
7.3 | IC50 | 4 | — | |
GKMMNQCWGZRQTN
|
7.3 | IC50 | 4 | — | |
JGQPZPLJOBHHBK
|
7.3 | IC50 | 3 | — | |
JHOCOFJBWLHCTN
|
7.3 | IC50 | 2 | — | |
JVAKWUYUZCOCKR
|
7.3 | IC50 | 4 | — | |
NTLLKKOHPKDCSW
|
7.3 | IC50 | 3 | — | |
OYMMHSBUFOLNEY
|
7.3 | IC50 | 3 | — | |
SOYMCIQWSHFMKE
|
7.3 | IC50 | 2 | — | |
ZJDRXPZROJHILR
|
7.3 | IC50 | 2 | — | |
JLNZMTDBARFXJN
|
7.3 | IC50 | 9 | — | |
BTGFLXGQPNRXDH
|
7.3 | IC50 | 3 | — | |
CAKYNETUOQZPMX
|
7.3 | IC50 | 2 | — | |
CBJPXYZHTAENCD
|
7.3 | IC50 | 2 | — | |
DNVXATUJJDPFDM
|
7.3 | IC50 | 2 | — | |
HSMCUAMXZNQLSQ
|
7.3 | IC50 | 3 | — | |
IMXDUOIANVGJIA
|
7.3 | IC50 | 3 | — | |
IMYHVLQAXUTNRG
|
7.3 | IC50 | 3 | — | |
PQSJCTLBPAPREX
|
7.3 | IC50 | 2 | — | |
WQEGQSRMXSLEON
|
7.3 | IC50 | 3 | — | |
AULNYQHQUIEHMG
|
7.3 | IC50 | 2 | — | |
BKQJIPRADVVRKL
|
7.3 | IC50 | 3 | — | |
HMXDNEFPCAGWPH
|
7.3 | IC50 | 3 | — | |
HZTRWCKQNKXISW
|
7.3 | Kd | 2 | — | |
OJGGGCDIKGWBSR
|
7.3 | IC50 | 2 | — | |
WOHDSOWPKUZJTL
|
7.3 | IC50 | 2 | — | |
BQZRFJLSVVFWBQ
|
7.3 | IC50 | 3 | — | |
HSYFXAZMBHUTJZ
|
7.3 | IC50 | 3 | — | |
LCWFKXOJTKLMHT
|
7.3 | IC50 | 2 | — | |
LCXHXIMNUYTCEI
|
7.3 | IC50 | 3 | — | |
LWGUCDPMTIPABX
|
7.3 | IC50 | 4 | — | |
QTVSDAUHDJBCAA
|
7.3 | IC50 | 4 | — | |
VLGYORZRSHEGRC
|
7.3 | IC50 | 2 | — | |
WODOTYIRVRGFSJ
|
7.3 | IC50 | 3 | — | |
XJKTXWSMMWPNTP
|
7.3 | IC50 | 6 | — | |
BQOVFHDJHUGBES
|
7.2 | IC50 | 2 | — | |
GQXFGAMRIGUNFT
|
7.2 | IC50 | 4 | — | |
HXGQYSSCVKIEIA
|
7.2 | IC50 | 3 | — | |
MZKIOOQWOZDDMX
|
7.2 | IC50 | 3 | — | |
OXYDGMKIFXNGOS
|
7.2 | IC50 | 3 | — |