Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ULIAHCSBBVNLGS
|
7.4 | IC50 | 3 | — | |
WPRFMKAORZZEIZ
|
7.4 | IC50 | 2 | — | |
WTDQWZPPVBDRKD
|
7.4 | IC50 | 3 | — | |
BALJMSOPRQWRAP
|
7.4 | IC50 | 3 | — | |
HDHIHYNEQCFQNL
|
7.4 | IC50 | 3 | — | |
IMBCMESWDHPIDA
|
7.4 | IC50 | 3 | — | |
UTSVADVXKCTABF
|
7.4 | IC50 | 3 | — | |
YTYPEASDFWXHLK
|
7.4 | IC50 | 3 | — | |
AREGGTVPTLNTCU
|
7.4 | IC50 | 3 | — | |
FMSBJUGTJUGWQX
|
7.4 | IC50 | 2 | — | |
IMXDUOIANVGJIA
|
7.4 | IC50 | 4 | — | |
IUUGMLRGSKSQJD
|
7.4 | IC50 | 3 | — | |
KBQLHGZSZFKGCG
|
7.4 | IC50 | 3 | — | |
LZYVFLZEQAANSW
|
7.4 | IC50 | 3 | — | |
WAEXFXRVDQXREF
|
7.4 | IC50 | 20 | Yes | |
WEWCBQWPGVKVPY
|
7.4 | IC50 | 2 | — | |
CYUUSRGILFWDHA
|
7.4 | IC50 | 2 | — | |
PBZMPCXVZAPRES
|
7.4 | IC50 | 3 | — | |
POKZINYHLOHGEB
|
7.4 | Kd | 4 | — | |
QXWJFGXUZLPVCL
|
7.4 | IC50 | 2 | — | |
QYUSWNWUSZFQJV
|
7.4 | IC50 | 2 | — | |
RKWOVOVDWBRGQO
|
7.4 | Kd | 5 | — | |
UCJMBWXOKLINTN
|
7.4 | IC50 | 4 | — | |
WYUJMOVTXOPUEX
|
7.4 | IC50 | 4 | — | |
XOEVAYXDSJABMS
|
7.4 | Ki | 3 | — | |
CJVJSGBELMMESS
|
7.3 | IC50 | 2 | — | |
CQPGVZBZRUVJJZ
|
7.3 | IC50 | 3 | — | |
GZEDEKFDZMUCGJ
|
7.3 | IC50 | 4 | — | |
OFWSNGJQSBQEOU
|
7.3 | IC50 | 2 | — | |
QLRYSHYUZMZZPY
|
7.3 | IC50 | 4 | — | |
STHZORHCRFBRIV
|
7.3 | IC50 | 3 | — | |
UFFMFBORABJCTA
|
7.3 | Ki | 3 | — | |
WKNJQMMPCXOMRN
|
7.3 | IC50 | 2 | — | |
XRQOPEVIGOZEJD
|
7.3 | IC50 | 3 | — | |
DAXLHHYYMDQRCH
|
7.3 | IC50 | 3 | — | |
IPNHNGIFOOJHDF
|
7.3 | IC50 | 3 | — | |
LMCSAEHKLPKZOO
|
7.3 | IC50 | 3 | — | |
SLTHVRXQOKFPLI
|
7.3 | IC50 | 3 | — | |
WAXXYIQBXWBHKY
|
7.3 | IC50 | 2 | — | |
XMZQWTVGYFDKCT
|
7.3 | IC50 | 2 | — | |
FTHLNVOKHACXIU
|
7.3 | IC50 | 3 | — | |
IFFAPYISKKZOPO
|
7.3 | IC50 | 4 | — | |
MBXHXEWZLTYTML
|
7.3 | IC50 | 3 | — | |
MDRXOFSNECSECW
|
7.3 | Ki | 3 | — | |
NJQDQDHZAAGIQX
|
7.3 | IC50 | 3 | — | |
WDUULYPCWOELII
|
7.3 | IC50 | 2 | — | |
YNMSRPUOAQPYLV
|
7.3 | IC50 | 3 | — | |
JFLRJPGRSNHGAL
|
7.3 | IC50 | 3 | — | |
KXQSVQUUJQXHIX
|
7.3 | IC50 | 2 | — | |
OCRZEXONTRGXJJ
|
7.3 | Kd | 3 | — |