Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OQBRSKHYDQIBJE
|
7.4 | IC50 | 3 | — | |
OYDMPDMTZYTSSQ
|
7.4 | IC50 | 3 | — | |
QNOJAPBYTXGBLX
|
7.4 | Ki | 5 | — | |
SMYPWBHABVYAJK
|
7.4 | IC50 | 3 | — | |
ZXGRKOXAZLNTEL
|
7.4 | IC50 | 2 | — | |
ZXGRKOXAZLNTEL
|
7.4 | IC50 | 2 | — | |
FFHFKSXIZXKTRE
|
7.4 | IC50 | 3 | — | |
HQEUJXGKBKBFIW
|
7.4 | IC50 | 3 | — | |
JNYUGWPUYNNZOZ
|
7.4 | Kd | 3 | — | |
PKFVMDLBSYTDCI
|
7.4 | IC50 | 2 | — | |
PPCFYGSMPQKDDM
|
7.4 | IC50 | 3 | — | |
PTCKKLKSUNCGCE
|
7.4 | Ki | 2 | — | |
SNDFCVARRAHINB
|
7.4 | IC50 | 3 | — | |
STGWRPISYALDEU
|
7.4 | IC50 | 2 | — | |
XQVVPGYIWAGRNI
|
7.4 | IC50 | 34 | — | |
IFLPDVNBLNGRJS
|
7.4 | IC50 | 3 | — | |
IPDBNDHFDHKHDZ
|
7.4 | IC50 | 3 | — | |
JHVSPUDTTXELLE
|
7.4 | IC50 | 3 | — | |
JUNKHWUBWMACDY
|
7.4 | IC50 | 3 | — | |
JVTTVFOTQZIFEV
|
7.4 | IC50 | 3 | — | |
PPMNCASBGOVBMV
|
7.4 | IC50 | 2 | — | |
RMSPJEQBXIFKPD
|
7.4 | IC50 | 3 | — | |
UHWNJFZTYJNBAN
|
7.4 | Kd | 5 | — | |
VLVRBRZAFGCGJV
|
7.4 | IC50 | 3 | — | |
AEOQRVQQPVQSRQ
|
7.4 | IC50 | 3 | — | |
CBNDXTMVECMPGV
|
7.4 | IC50 | 4 | — | |
DLEHIPJVRSZXAI
|
7.4 | Ki | 3 | — | |
FFMRDJNJHCWRIX
|
7.4 | IC50 | 3 | — | |
KOWPYSXWLGSRKS
|
7.4 | IC50 | 3 | — | |
NUBBUOMZQPTGKS
|
7.4 | IC50 | 2 | — | |
QGIHDISRDFTWAD
|
7.4 | IC50 | 3 | — | |
DNVXATUJJDPFDM
|
7.4 | IC50 | 4 | — | |
NEUUJGUKAZAFHZ
|
7.4 | IC50 | 3 | — | |
NMYGYOKYQBENRX
|
7.4 | IC50 | 2 | — | |
QIJUHAIEZZEKSX
|
7.4 | IC50 | 3 | — | |
QLRYSHYUZMZZPY
|
7.4 | IC50 | 3 | — | |
SCYDFQIUWZYQDE
|
7.4 | IC50 | 3 | — | |
UQMYMWRETIHSGQ
|
7.4 | IC50 | 3 | — | |
VUWJZAUOMZSUEU
|
7.4 | IC50 | 3 | — | |
YLTIAQHQEZGHPJ
|
7.4 | IC50 | 2 | — | |
ZJTYXGWJNWESQV
|
7.4 | Kd | 3 | — | |
ZORLJXWXFABTPZ
|
7.4 | IC50 | 9 | — | |
HKECFOZBEGKIAX
|
7.4 | IC50 | 3 | — | |
IISZWHJYEZSSQM
|
7.4 | IC50 | 2 | — | |
KIGOYJHUPSVEGZ
|
7.4 | IC50 | 2 | — | |
KTPZIQXMURKYQT
|
7.4 | IC50 | 2 | — | |
MUDFQCHHOJYXCS
|
7.4 | IC50 | 2 | — | |
NVRXYLMWFKVLJI
|
7.4 | IC50 | 3 | — | |
PYJQEIWIODYCRH
|
7.4 | IC50 | 3 | — | |
SJSCJYHUBPKPNG
|
7.4 | IC50 | 3 | — |