Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CJVJSGBELMMESS
|
7.5 | IC50 | 2 | — | |
CMEIUJXPMXIULZ
|
7.5 | IC50 | 3 | — | |
GYXAATIUVYEJQN
|
7.5 | IC50 | 3 | — | |
HTSUQACFQAFQAC
|
7.5 | IC50 | 2 | — | |
HXVCPXGIAZLACO
|
7.5 | IC50 | 2 | — | |
IENHPOBVKKOOQK
|
7.5 | IC50 | 2 | — | |
MMMRGZLSUKMQOD
|
7.5 | IC50 | 4 | — | |
MNDAWZZJIIHLSL
|
7.5 | IC50 | 2 | — | |
NBBLMCRKPAWOPH
|
7.5 | IC50 | 3 | — | |
OGJPTYDTRCDEJC
|
7.5 | IC50 | 3 | — | |
QWMJOPLEXJAKPN
|
7.5 | IC50 | 3 | — | |
WIFZFGUMQICZOO
|
7.5 | IC50 | 3 | — | |
WJAYJAKMQSJKDW
|
7.5 | IC50 | 3 | — | |
XZYFNQNYLMTZIS
|
7.5 | IC50 | 3 | — | |
FRMBPERTEITNRY
|
7.5 | IC50 | 2 | — | |
WHDUHJYPRJXLGF
|
7.5 | Kd | 4 | — | |
XOUGFEOTWVNPHI
|
7.5 | IC50 | 3 | — | |
AIPWZDCZUJGLIF
|
7.5 | IC50 | 3 | — | |
CURNKPOFSHNCQW
|
7.5 | IC50 | 2 | — | |
FAPXCSUYTUWYIY
|
7.5 | IC50 | 2 | — | |
GZFJPALDEYOFHA
|
7.5 | Ki | 6 | — | |
JBKUGHMRISDLDL
|
7.5 | IC50 | 3 | — | |
LVOINJWONMUWBO
|
7.5 | IC50 | 2 | — | |
PFPUXRWWYPANOO
|
7.5 | IC50 | 2 | — | |
QXTHZAMLLIIJHM
|
7.5 | IC50 | 3 | — | |
WAVOEVFKPHUSDB
|
7.5 | IC50 | 3 | — | |
WWFAGXVFIAJTJE
|
7.5 | IC50 | 2 | — | |
CDRNFZNHLRPDET
|
7.5 | IC50 | 2 | — | |
FMJBUHAFPYWEKA
|
7.5 | IC50 | 3 | — | |
IOHXSSTYGFWMFM
|
7.5 | IC50 | 3 | — | |
IVJMCRKXIOARPS
|
7.5 | IC50 | 3 | — | |
MQPRRCLCHOSXND
|
7.5 | IC50 | 3 | — | |
PXLJQXYHONWMKB
|
7.5 | IC50 | 3 | — | |
RGVADVPFHZUZFO
|
7.5 | IC50 | 2 | — | |
UOTPJXAROHNZGU
|
7.5 | IC50 | 2 | — | |
ZDYWXTGNQATUAC
|
7.5 | IC50 | 2 | — | |
AURWSPRKUDZZIW
|
7.5 | IC50 | 3 | — | |
DNVXATUJJDPFDM
|
7.5 | IC50 | 4 | — | |
IXNBIPCXYOBMSS
|
7.5 | IC50 | 3 | — | |
KOYGJJMRJVPCNS
|
7.5 | IC50 | 3 | — | |
OABQDWQBXSGEDG
|
7.5 | IC50 | 9 | — | |
SUFVOUWYHJXPBW
|
7.5 | Kd | 4 | — | |
WPRFMKAORZZEIZ
|
7.5 | IC50 | 3 | — | |
XQGQHZQHQKHLDK
|
7.5 | IC50 | 3 | — | |
ZSBDKRBBDNFMHY
|
7.5 | Ki | 3 | — | |
ZSHUBSUFZWWFGQ
|
7.5 | IC50 | 2 | — | |
FRVZZHQYKGFUEH
|
7.4 | IC50 | 2 | — | |
HSMCUAMXZNQLSQ
|
7.4 | IC50 | 3 | — | |
HZOZVQZXYYKRSX
|
7.4 | IC50 | 2 | — | |
OHRURASPPZQGQM
|
7.4 | IC50 | 14 | — |