Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTOVUBXMOLCWFF
|
7.6 | IC50 | 2 | — | |
BSZDTJJAUVZTBS
|
7.5 | IC50 | 3 | — | |
BYHXJJUONGOTKC
|
7.5 | IC50 | 2 | — | |
FLEGAAQBQHISDY
|
7.5 | IC50 | 3 | — | |
GJZVZCJWTFBXDP
|
7.5 | IC50 | 2 | — | |
HTPNGOWITIWAHM
|
7.5 | IC50 | 3 | — | |
MVAYDDZVYGANLI
|
7.5 | IC50 | 3 | — | |
RWLOGRLTDKDANT
|
7.5 | Kd | 2 | — | |
UHWGSUFICDUCKV
|
7.5 | IC50 | 3 | — | |
VVSCZWKYDATSNC
|
7.5 | IC50 | 3 | — | |
WQEGQSRMXSLEON
|
7.5 | IC50 | 4 | — | |
ZKVURPUQVABYSC
|
7.5 | IC50 | 3 | — | |
ZXGRKOXAZLNTEL
|
7.5 | IC50 | 2 | — | |
ZXGRKOXAZLNTEL
|
7.5 | IC50 | 2 | — | |
FQEWVABJRCOJBI
|
7.5 | IC50 | 4 | — | |
GKJNYZBASPYBEP
|
7.5 | IC50 | 3 | — | |
GVCFSBGCJBRHFS
|
7.5 | IC50 | 4 | — | |
JADOFDPLHYUWBU
|
7.5 | IC50 | 3 | — | |
NHMJYXDPZTZGQX
|
7.5 | IC50 | 2 | — | |
NHMJYXDPZTZGQX
|
7.5 | IC50 | 2 | — | |
PIKWYDHWUKSWAQ
|
7.5 | Kd | 4 | — | |
UCOMAESNVXJEIJ
|
7.5 | IC50 | 2 | — | |
UCTNVNGRNJPSOM
|
7.5 | IC50 | 3 | — | |
VFDAORCFAAAXRV
|
7.5 | IC50 | 3 | — | |
LNIICUXUOAFIAD
|
7.5 | IC50 | 12 | — | |
ZJKGEINLDGYOLW
|
7.5 | IC50 | 2 | — | |
FKGDRMFOMMYLPA
|
7.5 | IC50 | 3 | — | |
FRJGKZLDWJMCPQ
|
7.5 | IC50 | 3 | — | |
GTOKRJQCMDFUOW
|
7.5 | IC50 | 2 | — | |
IKKUVCXGUJTONF
|
7.5 | IC50 | 6 | — | |
JKTAXQJDSRMHSS
|
7.5 | IC50 | 3 | — | |
MVAYDDZVYGANLI
|
7.5 | IC50 | 3 | — | |
OTKIKJDBYKBEOE
|
7.5 | IC50 | 3 | — | |
PHSQIKIQGFDDEU
|
7.5 | IC50 | 2 | — | |
RKSYSKOBHCWHKB
|
7.5 | IC50 | 3 | — | |
SNXGAWWAXJMADO
|
7.5 | IC50 | 3 | — | |
UCBSOBAEFNVYID
|
7.5 | IC50 | 2 | — | |
WODOTYIRVRGFSJ
|
7.5 | IC50 | 3 | — | |
XNRZMTWJFLFRMR
|
7.5 | IC50 | 4 | — | |
XTZPTYMYXVFWJT
|
7.5 | IC50 | 3 | — | |
XYESNEVBCXKVML
|
7.5 | IC50 | 2 | — | |
ZUEZEQZVGBUYFN
|
7.5 | IC50 | 3 | — | |
AXKZAOMIZYICQV
|
7.5 | IC50 | 2 | — | |
FRDRCUWLVRNFIJ
|
7.5 | IC50 | 3 | — | |
GKMMNQCWGZRQTN
|
7.5 | IC50 | 2 | — | |
NCEJUIVQBWZGMA
|
7.5 | IC50 | 3 | — | |
PBHCWSGBMHUVGJ
|
7.5 | IC50 | 2 | — | |
SYJHORXMXBZSSH
|
7.5 | IC50 | 3 | — | |
WUFYDWKEOKQEEP
|
7.5 | IC50 | 3 | — | |
YTKVHFHJCRSLOJ
|
7.5 | IC50 | 2 | — |