Target Details
| UniProt AC | O60885 |
|---|---|
| Gene Symbol | BRD4 |
| Protein Name | Bromodomain-containing protein 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF17105 (BRD4_CDT) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 1,567
- Clinical molecules 4
- Avg pChEMBL 7.15
Associated Diseases (1)
Active Molecules (1,567)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FZWPGKYEENZFAU
|
10.9 | Kd | 4 | — | |
OPVRCPHGQNNHNN
|
10.8 | Kd | 2 | — | |
KYCQRWFJRCYKBU
|
10.6 | Kd | 2 | — | |
WHJGVHRMVTVKHR
|
10.6 | Kd | 2 | — | |
YQUPOPCILRFMSA
|
10.5 | Kd | 2 | — | |
NOYKJWSXDSTVCB
|
10.3 | Kd | 2 | — | |
JNSLBXJNVHYNNW
|
10.1 | Ki | 4 | — | |
VGOFJMULWAVDMV
|
9.5 | Kd | 2 | — | |
AIWLOFZSVQLGOB
|
9.4 | IC50 | 2 | — | |
LDUXKZCPPPHDPU
|
9.4 | IC50 | 2 | — | |
OMGCJTKEQJWTOY
|
9.3 | IC50 | 2 | — | |
HBOUBVJSLHNSNT
|
9.3 | IC50 | 2 | — | |
LHUPUFVIXSYKRE
|
9.2 | IC50 | 2 | — | |
OPGYUCHNVCWIIN
|
9.2 | IC50 | 2 | — | |
YYKFSJHHADBYMX
|
9.2 | IC50 | 2 | — | |
IUZLBZYYGQFQJZ
|
9.2 | IC50 | 2 | — | |
LMLIBNUOIWAJFC
|
9.1 | IC50 | 9 | — | |
UJARZGSRRXPOTK
|
9.1 | IC50 | 3 | — | |
UJARZGSRRXPOTK
|
9.1 | IC50 | 3 | — | |
DBKJPAGKXDFFCG
|
9.0 | IC50 | 2 | — | |
KAGYLLHUHGBNTA
|
9.0 | IC50 | 2 | — | |
KAYFVHVSQSDACO
|
9.0 | IC50 | 2 | — | |
KECYVMVFYPBARC
|
9.0 | IC50 | 2 | — | |
OPRLJTKXGDBVAC
|
9.0 | IC50 | 2 | — | |
PMNZVZQYPSMXDO
|
9.0 | IC50 | 2 | — | |
PSFDBOWKEFILAQ
|
9.0 | IC50 | 2 | — | |
RWUFFMJUVGICHP
|
9.0 | IC50 | 2 | — | |
XUGFYFHLYOPQJS
|
9.0 | IC50 | 2 | — | |
YPPIBRNYHDEWID
|
9.0 | IC50 | 2 | — | |
AXQYYKHQHMDBFK
|
9.0 | IC50 | 2 | — | |
KGERZPVQIRYWRK
|
9.0 | IC50 | 4 | — | |
AIWLOFZSVQLGOB
|
8.9 | IC50 | 2 | — | |
LJLJARSDBHJRGG
|
8.9 | Ki | 4 | — | |
UNODBAFOZVBZBF
|
8.8 | Ki | 4 | — | |
VLYMRIROHVATMC
|
8.8 | Kd | 2 | — | |
XCLRZZASCPTRLU
|
8.8 | IC50 | 2 | — | |
LZAPXWCSDTYFNB
|
8.7 | IC50 | 3 | — | |
PHSKNIAWTPPDAY
|
8.7 | IC50 | 2 | — | |
BKOMFGNROQEUHF
|
8.7 | IC50 | 2 | — | |
CUAGRANTRNSGSF
|
8.7 | IC50 | 2 | — | |
DFHREBKXJWXHKG
|
8.7 | Kd | 2 | — | |
DJNGAENPUAKERE
|
8.7 | IC50 | 2 | — | |
FMFGVLUVPAHDDT
|
8.7 | IC50 | 2 | — | |
FOLIJXOPRUSFGM
|
8.7 | IC50 | 2 | — | |
HPXHQNWBKFNTMR
|
8.7 | IC50 | 2 | — | |
HSOYPKXYVCVZOK
|
8.7 | IC50 | 2 | — | |
ICKGOXSYBTWKAP
|
8.7 | IC50 | 2 | — | |
JIYPVUCBRQNICX
|
8.7 | Kd | 7 | — | |
KRAIKLYQMMJWDD
|
8.7 | IC50 | 2 | — | |
NGRKNMYUPWAPCQ
|
8.7 | IC50 | 2 | — |