Target Details
| UniProt AC | O60755 |
|---|---|
| Gene Symbol | GALR3 |
| Protein Name | Galanin receptor type 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 25
- Clinical molecules 0
- Avg pChEMBL 7.17
KEGG Pathways (1)
Active Molecules (25)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HXCJZIBJTFITNI
|
8.3 | Ki | 3 | — | |
XNHSIZYARJUIGK
|
8.2 | Ki | 3 | — | |
DWFZBUWUXWZWKD
|
8.2 | IC50 | 4 | — | |
SLZIZIJTGAYEKK
|
8.0 | Ki | 3 | — | |
HTINXISERLHZAZ
|
7.9 | Ki | 3 | — | |
JWMXJVFGTXYBFM
|
7.8 | Kd | 3 | — | |
TXCGMRVPXUBHAL
|
7.8 | Ki | 2 | — | |
AHGJZJCKZYITJQ
|
7.7 | Ki | 2 | — | |
DTFARBHXORYQBF
|
7.4 | IC50 | 2 | — | |
TZOJVPDIYKRJSM
|
7.4 | Kd | 3 | — | |
VQUPYGXNBXITAA
|
7.4 | Ki | 3 | — | |
WGWNRQMTUPJGCW
|
7.2 | Ki | 3 | — | |
CBSXZYWGVAQSHI
|
7.2 | Ki | 3 | — | |
YWWOWEJNZKADMM
|
7.2 | Kd | 3 | — | |
XHARTEHOSRSMSF
|
7.1 | IC50 | 4 | — | |
WYBZIJBKCXMOCE
|
6.9 | IC50 | 2 | — | |
WEZRHPWWPXDLTL
|
6.8 | IC50 | 3 | — | |
CIEDGRWWCWXCMK
|
6.8 | IC50 | 3 | — | |
GXLKSVCDXUMIAV
|
6.6 | IC50 | 3 | — | |
OSGCBUDLRBUEGW
|
6.5 | Ki | 3 | — | |
FHTSPMGFAZMZJT
|
6.5 | Kd | 3 | — | |
OIPILFWXSMYKGL
|
6.2 | IC50 | 6 | — | |
LDEAEHIIHOWDLI
|
6.0 | Ki | 3 | — | |
NUGXOOKVHNJHDS
|
6.0 | Ki | 3 | — | |
XZOKDXWQSCIKCM
|
6.0 | IC50 | 2 | — |