Target Details
| UniProt AC | O60741 |
|---|---|
| Gene Symbol | HCN1 |
| Protein Name | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF08412 (Ion_trans_N) |
Summary
- Multi-target molecules 10
- Clinical molecules 0
- Avg pChEMBL 6.98
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQURIRADMQBJKA
|
7.8 | IC50 | 2 | — | |
ICQOHPXXADVTOI
|
7.5 | IC50 | 2 | — | |
YGTKBUSFMKESCS
|
7.5 | IC50 | 2 | — | |
NZCJBWNCSCYPKE
|
7.3 | IC50 | 2 | — | |
GKHQMAHQZSEGLJ
|
7.1 | IC50 | 2 | — | |
JABSKGQQWUDVRU
|
6.8 | IC50 | 2 | — | |
JHYUXYFUZXQBNW
|
6.7 | IC50 | 2 | — | |
IQBSKXRURIYRNZ
|
6.4 | IC50 | 2 | — | |
LFDSRDSBKYSENL
|
6.4 | IC50 | 2 | — | |
QVVGKUPYQMYUFR
|
6.3 | IC50 | 2 | — |