Target Details
| UniProt AC | O60678 |
|---|---|
| Gene Symbol | PRMT3 |
| Protein Name | Protein arginine N-methyltransferase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21137 (ANM3_C2H2_Zf) PF21336 (ANM3_zf-C2H2) PF06325 (PrmA) PF22528 (PRMT_C) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 6.8
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SPEGERVLTUWZPA
|
8.8 | IC50 | 5 | — | |
XCZUYGFLWBJNCB
|
7.7 | IC50 | 4 | — | |
FMTVWAGUJRUAKE
|
7.3 | IC50 | 5 | — | |
LUBCTIQAZDQPJR
|
6.9 | IC50 | 5 | — | |
ZJUKTBDSGOFHSH
|
6.5 | IC50 | 22 | — | |
CBLOJJICRSGZRU
|
6.5 | IC50 | 4 | — | |
DVZZYZNFLHFCPI
|
6.5 | IC50 | 7 | — | |
CNMWTZSRTFSQJJ
|
6.3 | IC50 | 5 | — | |
VZDPLMKEFMWBMM
|
6.3 | Ki | 5 | — | |
XLTWYAYAFLGUEQ
|
6.1 | IC50 | 3 | — | |
UMKLFWMQTDMELK
|
6.0 | IC50 | 5 | — |