Target Details
UniProt ACO60674
Gene SymbolJAK2
Protein NameTyrosine-protein kinase JAK2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF18379 (FERM_F1) PF18377 (FERM_F2) PF17887 (Jak1_Phl) PF07714 (PK_Tyr_Ser-Thr) PF21990 (SH2_1)
Summary
  • Multi-target molecules 10,545
  • Clinical molecules 78
  • Avg pChEMBL 7.81
Top Co-occurrence Targets
Active Molecules (10,545)
InChIKey pChEMBL Type Targets Clinical
ZFIYENYHDMNREK 9.7 Ki 2
CZCGCTUNTFUHHU 9.7 IC50 4
YYUFVSMURUQLMO 9.7 IC50 4
ADMZIYBQCUQEFO 9.7 Ki 2
BWGLFRJYQLOIII 9.7 Ki 2
CAHYIXKHAUSRRA 9.7 IC50 2
DKFMXHXDTZQTJB 9.7 IC50 2
FOPMKMPCLCPQTK 9.7 IC50 2
KXUAMYAVSZHGDY 9.7 IC50 2
KYQCJGPWKAIKCS 9.7 Ki 4
LNDOFTXPTPMZBR 9.7 IC50 2
LZRZLWVRSQYJDT 9.7 IC50 2
MTNOHNLEHSEDJU 9.7 IC50 2
NIVDAFZUMYCAFE 9.7 Ki 2
ODDNPGSYZFWGMF 9.7 IC50 2
QGKIINSCKDFRPR 9.7 Ki 4
SFJVTTMWKMNHQE 9.7 IC50 2
SGSAHEBNHCGXMY 9.7 Ki 2
SPBXVFLBMBIHKF 9.7 Ki 2
SRNCIGCIBSHWSA 9.7 Ki 2
VBIIHZOALUSRNV 9.7 IC50 4
AFWJENUAHKAUTF 9.7 IC50 4
JIQQEQXPBPQIPX 9.7 IC50 4
RFBZHSXCSARQJM 9.7 Ki 2
ADCNRVPERNLLDX 9.7 Ki 2
AEYXDCFBNVYPGT 9.7 Ki 2
BGLUIKXULQMNGE 9.7 IC50 2
CMQVWDQTOHJZLK 9.7 IC50 2
DRLOGZHQVDXOPP 9.7 IC50 2
DYBLTFRYGJITIL 9.7 Ki 2
GJEFXVFPINXVME 9.7 IC50 2
GSLRMDBWPNBYFD 9.7 Ki 2
GXUMCSNXFVXLMX 9.7 IC50 2
HHPOPPAYAQSYTK 9.7 Ki 2
IATRTMWSBYEFLC 9.7 Ki 2
KWGLHLYWTQSATC 9.7 IC50 3
LBBZLXMPUULIGG 9.7 IC50 2
LOUVYDGMLXYULX 9.7 Ki 2
MBBKLMHHKNIWTK 9.7 Ki 2
MTAYQODFZKDBIN 9.7 Ki 2
NRQSCGVAXSQZCR 9.7 IC50 4
QLZHYINEOIHHAY 9.7 Ki 2
QQZRLGYOWDXZII 9.7 Ki 2
TWGKDJAUEJWZFH 9.7 IC50 2
TWGKDJAUEJWZFH 9.7 IC50 2
VKERTUOBZIKJDO 9.7 Ki 2
YENOZGNVRCRNCQ 9.7 Ki 4
YLAKIDRGVDYWAA 9.7 IC50 2
YZMIQTVIZUMJRU 9.7 Ki 2
ZMFNZTSECWNPOO 9.7 IC50 2
2D structure