Target Details
| UniProt AC | O60658 |
|---|---|
| Gene Symbol | PDE8A |
| Protein Name | High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00989 (PAS) PF08629 (PDE8) PF23198 (PDE8A_N) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 25
- Clinical molecules 0
- Avg pChEMBL 8.04
KEGG Pathways (5)
Active Molecules (25)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJLHNYPXKZJKLV
|
10.0 | IC50 | 24 | — | |
KXCOKRBRUWINCT
|
9.9 | IC50 | 24 | — | |
KPFFPWNKWSYQFT
|
9.8 | IC50 | 24 | — | |
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
VNLPYEMGHGDRRZ
|
9.2 | IC50 | 2 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
FIUCLBJMUGCQTF
|
9.0 | IC50 | 8 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
DWHZRFMVWCPXSM
|
8.7 | IC50 | 2 | — | |
KTZOPPLFULGANJ
|
8.7 | IC50 | 2 | — | |
WZGVFBPGGTVOPK
|
8.7 | IC50 | 2 | — | |
QGTJGTFOISKMAD
|
8.7 | IC50 | 2 | — | |
ORTHDXKTDAKOBP
|
7.8 | IC50 | 3 | — | |
JYHQBYXSPOBQMT
|
6.8 | IC50 | 3 | — | |
ZMZGFAGXALOLIK
|
6.7 | IC50 | 4 | — | |
INDKHRIZOIEPIG
|
6.5 | IC50 | 2 | — | |
OFZGCAMFVYIIHV
|
6.5 | IC50 | 24 | — | |
BBHYMAIPZZCFDD
|
6.4 | IC50 | 3 | — | |
IZEKFCXSFNUWAM
|
6.3 | IC50 | 19 | — | |
IWQJRWQPBCCRGZ
|
6.2 | IC50 | 8 | — | |
OVSHRJGAYOZGQR
|
6.2 | IC50 | 8 | — | |
IOKJCBWLGAJZFW
|
6.1 | IC50 | 2 | — | |
JITUOVWOCIXEEZ
|
6.0 | IC50 | 23 | — |